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Found 237 with Last Name = 'koike' and Initial = 'k'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213889(3-[(Z)-5,6,7,8-tetrahydro-naphthalen-1-ylimino]-2-...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503606(CHEMBL4462756)
Affinity DataKi:  0.620nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256379(CHEMBL482356 | methyl 3-(4-chloronaphthalen-1-ylim...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to mouse CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213889(3-[(Z)-5,6,7,8-tetrahydro-naphthalen-1-ylimino]-2-...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256378(CHEMBL482355 | methyl 3-(4-fluoronaphthalen-1-ylim...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213881(3-[(Z)-2-isopropyl-phenylimino]-2-thia-4-aza-spiro...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256379(CHEMBL482356 | methyl 3-(4-chloronaphthalen-1-ylim...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256218(CHEMBL516406 | methyl 3-(naphthalen-1-ylimino)-2-o...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256318(CHEMBL481508 | methyl 3-(3-tert-butylisoxazol-5-yl...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213900(3-[(Z)-benzo[1,2,5]oxadiazol-4-ylimino]-2-thia-4-a...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256315(CHEMBL469895 | methyl 3-(2-methoxyphenylimino)-2-o...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503604(Naldemedine | S-297995)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503597(CHEMBL4534307)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256317(CHEMBL511790 | methyl 3-(4-tert-butylthiazol-2-yli...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256319(CHEMBL519288 | methyl 3-(3-(3-ethylpentan-3-yl)iso...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213891(3-[(Z)-3-methoxy-phenylimino]-2-thia-4-aza-spiro[5...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256319(CHEMBL519288 | methyl 3-(3-(3-ethylpentan-3-yl)iso...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213888(8-[(Z)-2-isopropyl-phenylimino]-7-thia-9-aza-spiro...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213883(3-[(Z)-2,3-dimethyl-phenylimino]-2-thia-4-aza-spir...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256318(CHEMBL481508 | methyl 3-(3-tert-butylisoxazol-5-yl...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503611(CHEMBL4468216)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503601(CHEMBL4529950)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256317(CHEMBL511790 | methyl 3-(4-tert-butylthiazol-2-yli...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256431(CHEMBL480578 | methyl 3-(5,6,7,8-tetrahydronaphtha...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213893(3-[(Z)-1-methyl-1,2,3,4-tetrahydro-quinolin-5-ylim...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503604(Naldemedine | S-297995)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213885(3-[(Z)-2-trifluoromethyl-phenylimino]-2-thia-4-aza...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503596(CHEMBL4561876)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213899(3-[(Z)-2-methoxy-phenylimino]-2-thia-4-aza-spiro[5...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213904(3-[(Z)-4-ethyl-phenylimino]-2-thia-4-aza-spiro[5.5...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213881(3-[(Z)-2-isopropyl-phenylimino]-2-thia-4-aza-spiro...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to mouse CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503599(CHEMBL4439770)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213884(3-[(Z)-benzo[1,2,5]thiadiazol-4-ylimino]-2-thia-4-...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503598(CHEMBL4551066)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256219(CHEMBL475772 | S-methyl 3-(naphthalen-1-ylimino)-2...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM102406(US8536192, I-135)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256380(CHEMBL482357 | methyl 3-(4-cyanonaphthalen-1-ylimi...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256433(CHEMBL481888 | methyl 3-(4-cyano-5,6,7,8-tetrahydr...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503600(CHEMBL4542825)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503610(CHEMBL4516674)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213887(3-[(Z)-4-cyano-phenylimino]-2-thia-4-aza-spiro[5.5...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256381(CHEMBL519635 | methyl 3-(4-nitronaphthalen-1-ylimi...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503594(CHEMBL4574150)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213897(3-[(Z)-3-isopropyl-phenylimino]-2-thia-4-aza-spiro...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503600(CHEMBL4542825)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50256379(CHEMBL482356 | methyl 3-(4-chloronaphthalen-1-ylim...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity to human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50213901(3-[(Z)-4-methoxy-phenylimino]-2-thia-4-aza-spiro[5...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503607(CHEMBL4452187)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu-opioid receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50503612(CHEMBL4459343)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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