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Found 260 with Last Name = 'kopcho' and Initial = 'lm'
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119489(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi:  4nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119488(CHEMBL143628 | X1-(4-Chloro-phenyl)-1H-pyrazole-3,...)
Affinity DataKi:  4nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119481(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi:  6nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119483(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi:  8nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119485(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  12nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119490(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  26nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119492(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi:  32nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119487(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi:  91nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119491(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  138nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119484(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  331nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119482(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119486(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of dihydroorotate dehydrogenase (DHODase) of Helicobacter pyloriMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119485(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119484(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119486(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119491(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119487(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119490(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119489(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119488(CHEMBL143628 | X1-(4-Chloro-phenyl)-1H-pyrazole-3,...)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119483(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119492(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119481(1-(4-Chloro-phenyl)-1H-pyrazole-3,5-dicarboxylic a...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50119482(1-(4-Methoxy-phenyl)-1H-pyrazole-3,5-dicarboxylic ...)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human dihydroorotate dehydrogenase (DHODase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatic triacylglycerol lipase(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50525871(CHEMBL4460999)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of hepatic lipase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50525871(CHEMBL4460999)
Affinity DataIC50:  1nMAssay Description:Inhibition of endothelial lipase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50554034(CHEMBL4747269)
Affinity DataIC50:  1nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 120 mM NaCl by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50554035(CHEMBL4790231)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 120 mM NaCl by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50554052(CHEMBL4763667)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 120 mM NaCl by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50554050(CHEMBL4752248)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 120 mM NaCl by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50554057(CHEMBL4740830)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 120 mM NaCl by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50525879(CHEMBL4541404)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of endothelial lipase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHepatic triacylglycerol lipase(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50525869(CHEMBL4587475)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of hepatic lipase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50554056(CHEMBL4782307)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 120 mM NaCl by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50554054(CHEMBL4751166)
Affinity DataIC50:  9.30nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 120 mM NaCl by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50525869(CHEMBL4587475)
Affinity DataIC50:  13nMAssay Description:Inhibition of endothelial lipase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50552364(CHEMBL4781606)
Affinity DataIC50:  14nMAssay Description:Displacement of fluorescent labeled probe from human recombinant His-tagged TNFalpha (77 to 233 residues) expressed in Escherichia coli preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50552381(CHEMBL4787433)
Affinity DataIC50:  15nMAssay Description:Displacement of fluorescent labeled probe from human recombinant His-tagged TNFalpha (77 to 233 residues) expressed in Escherichia coli preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50552380(CHEMBL4797699)
Affinity DataIC50:  15nMAssay Description:Displacement of fluorescent labeled probe from human recombinant His-tagged TNFalpha (77 to 233 residues) expressed in Escherichia coli preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50525868(CHEMBL4557646)
Affinity DataIC50:  15nMAssay Description:Inhibition of endothelial lipase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50554051(CHEMBL4795827)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 120 mM NaCl by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50525878(CHEMBL4581408)
Affinity DataIC50:  16nMAssay Description:Inhibition of endothelial lipase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM357630(7-(3- chlorobenzyl)- 3H- [1,2,3]triazolo [4,5-b]py...)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 240 mM NaCl and 10 uM H2O2 by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50554036(CHEMBL4764237)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins by amplex red dye based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM357653(3-((5-amino- 3H- [1,2,3]triazolo [4,5-b] pyridin- ...)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 240 mM NaCl and 10 uM H2O2 by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50552368(CHEMBL4787001)
Affinity DataIC50:  17nMAssay Description:Displacement of fluorescent labeled probe from human recombinant His-tagged TNFalpha (77 to 233 residues) expressed in Escherichia coli preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMyeloperoxidase(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50554055(CHEMBL4755252)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant human MPO incubated for 10 mins in presence of 120 mM NaCl by aminophenyl fluorescein based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50552388(CHEMBL4742065)
Affinity DataIC50:  24nMAssay Description:Displacement of fluorescent labeled probe from human recombinant His-tagged TNFalpha (77 to 233 residues) expressed in Escherichia coli preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50552388(CHEMBL4742065)
Affinity DataIC50:  24nMAssay Description:Displacement of fluorescent labeled probe from human recombinant His-tagged TNFalpha (77 to 233 residues) expressed in Escherichia coli preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50552388(CHEMBL4742065)
Affinity DataIC50:  24nMAssay Description:Displacement of fluorescent labeled probe from human recombinant His-tagged TNFalpha (77 to 233 residues) expressed in Escherichia coli preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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