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Found 71 with Last Name = 'koshizawa' and Initial = 't'
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50094851(CHEMBL3589803)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50172720(CHEMBL3814017)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50172721(CHEMBL3814026)
Affinity DataEC50:  860nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50173929(CHEMBL3814025)
Affinity DataEC50:  1.96E+3nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50174995(CHEMBL3814000)
Affinity DataEC50:  2.89E+3nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50176997(CHEMBL3814071)
Affinity DataEC50:  3.14E+3nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179403(CHEMBL3814381)
Affinity DataEC50:  360nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179430(CHEMBL3813703)
Affinity DataEC50:  400nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179431(CHEMBL3814351)
Affinity DataEC50:  3.74E+3nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179484(CHEMBL3814980)
Affinity DataEC50:  340nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179485(CHEMBL3814799)
Affinity DataEC50:  330nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179485(CHEMBL3814799)
Affinity DataEC50:  330nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataEC50:  490nMAssay Description:Agonist activity at GAL4 fused LXRalpha (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50064330(CHEMBL3403710)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50094851(CHEMBL3589803)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50172720(CHEMBL3814017)
Affinity DataEC50:  800nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50172721(CHEMBL3814026)
Affinity DataEC50:  610nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50173929(CHEMBL3814025)
Affinity DataEC50:  500nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179486(CHEMBL3814224)
Affinity DataEC50:  1.81E+3nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50174995(CHEMBL3814000)
Affinity DataEC50:  2.85E+3nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179488(CHEMBL3814807)
Affinity DataEC50:  1.88E+3nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50176997(CHEMBL3814071)
Affinity DataEC50:  700nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179489(CHEMBL3814297)
Affinity DataEC50:  1.66E+3nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179490(CHEMBL3813961)
Affinity DataEC50:  2.87E+3nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179491(CHEMBL3814806)
Affinity DataEC50:  2.33E+3nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179403(CHEMBL3814381)
Affinity DataEC50:  120nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179430(CHEMBL3813703)
Affinity DataEC50:  64nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179431(CHEMBL3814351)
Affinity DataEC50:  360nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179484(CHEMBL3814980)
Affinity DataEC50:  110nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179485(CHEMBL3814799)
Affinity DataEC50:  58nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179485(CHEMBL3814799)
Affinity DataEC50:  58nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50179485(CHEMBL3814799)
Affinity DataEC50:  7nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataEC50:  410nMAssay Description:Agonist activity at GAL4 fused LXRbeta-LBD (unknown origin) transfected in CHOK1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268607(CHEMBL4060970)
Affinity DataEC50:  793nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268608(CHEMBL4072360)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268613(CHEMBL4099307)
Affinity DataEC50:  53nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268614(CHEMBL4098382)
Affinity DataEC50:  129nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268615(CHEMBL4065753)
Affinity DataEC50:  353nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268617(CHEMBL4093367)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268618(CHEMBL4083015)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268619(CHEMBL4100997)
Affinity DataEC50:  79nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268621(CHEMBL4101938)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268622(CHEMBL4077670)
Affinity DataEC50:  201nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268623(CHEMBL4063942)
Affinity DataEC50:  310nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268624(CHEMBL4085517)
Affinity DataEC50:  391nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268630(CHEMBL4086445)
Affinity DataEC50:  586nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268631(CHEMBL4104336)
Affinity DataEC50:  78nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268637(CHEMBL4094202)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells co-expressing CRE-luciferase incubated for 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268638(CHEMBL4080356)
Affinity DataEC50:  82nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Kowa

Curated by ChEMBL
LigandPNGBDBM50268639(CHEMBL4099566)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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