TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 2.00E+4nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 2.80E+4nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 4.10E+4nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 5.40E+4nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 5.60E+4nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 8.00E+4nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 8.10E+4nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 9.60E+4nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.10E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.10E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.50E+5nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.60E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.70E+5nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.90E+5nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 2.00E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 2.10E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 2.10E+5nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 2.50E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 2.60E+5nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+5nMAssay Description:Inhibition of human serine racemaseMore data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 3.60E+5nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 3.89E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 4.30E+5nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 4.90E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 5.00E+5nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 5.50E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 5.70E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
Affinity DataKi: 6.10E+5nMAssay Description:Inhibition of human serine racemaseMore data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 7.60E+5nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAminodeoxychorismate lyase(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 7.70E+5nMAssay Description:Inhibition of Escherichia coli K12 ADCS by spectrophotometryMore data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 7.90E+5nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetAminodeoxychorismate lyase(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of Escherichia coli K12 ADCS by spectrophotometryMore data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.02E+6nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.08E+6nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.20E+6nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 1.30E+6nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetAminodeoxychorismate lyase(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 2.50E+6nMAssay Description:Inhibition of Escherichia coli K12 ADCS by spectrophotometryMore data for this Ligand-Target Pair
TargetAnthranilate synthase component 1(Salmonella typhimurium)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 2.60E+6nMAssay Description:Inhibition of Salmonella typhimurium anthranilate synthase trpE:trpD expressed in Escherichia coli BL21(DE3) coexpressing stop codon in trpD gene for...More data for this Ligand-Target Pair
TargetIsochorismate synthase EntC(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 2.60E+6nMAssay Description:Inhibition of Escherichia coli K12 IS expressed in Escherichia coli BL21(DE3) by spectrophotometryMore data for this Ligand-Target Pair
TargetAminodeoxychorismate lyase(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 5.70E+6nMAssay Description:Inhibition of Escherichia coli K12 ADCS by spectrophotometryMore data for this Ligand-Target Pair
TargetAminodeoxychorismate lyase(Escherichia coli (strain K12))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 6.80E+6nMAssay Description:Inhibition of Escherichia coli K12 ADCS by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0370nMAssay Description:Inhibition of human integrin alpha-4-beta-1-mediated MOLT4 cell adhesion to biotin-conjugated CS-1 peptideMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0372nMpH: 7.5 T: 2°CAssay Description:Binding affinities (IC50) of the ligands were studied in a Molt-4 T-cell adhesion assay by inhibiting the alpha-4/beta-1 mediated cell adhesion to CS...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0530nMAssay Description:Inhibition of human integrin alpha-4-beta-1-mediated MOLT4 cell adhesion to biotin-conjugated CS-1 peptideMore data for this Ligand-Target Pair
Affinity DataIC50: 0.305nMpH: 7.5 T: 2°CAssay Description:Binding affinities (IC50) of the ligands were studied in a Molt-4 T-cell adhesion assay by inhibiting the alpha-4/beta-1 mediated cell adhesion to CS...More data for this Ligand-Target Pair
Affinity DataIC50: 0.305nMAssay Description:Inhibition of human integrin alpha-4-beta-1-mediated MOLT4 cell adhesion to biotin-conjugated CS-1 peptideMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human integrin alpha-4-beta-1-mediated MOLT4 cell adhesion to biotin-conjugated CS-1 peptideMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of wild type human CFTR chloride conductance expressed in forskolin-stimulated rat FRT cells by short-circuit current analysis in presence...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human integrin alpha-4-beta-1-mediated MOLT4 cell adhesion to biotin-conjugated CS-1 peptideMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells assessed as inhibition of forskolin-induced short-circuit current by voltage clamp electrop...More data for this Ligand-Target Pair