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Found 45 with Last Name = 'kusama' and Initial = 'h'
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198353(CHEMBL227753 | CHEMBL534948 | N-(2,6-dimethylpheny...)
Affinity DataIC50:  8nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198360(CHEMBL227906 | N-(2,6-dimethylphenyl)-5-(3-methoxy...)
Affinity DataIC50:  11nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198372(CHEMBL387641 | N-(2,6-dimethylphenyl)-5-thiophen-2...)
Affinity DataIC50:  12nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198370(CHEMBL223873 | N-(2,6-dimethyl-phenyl)-5-phenylimi...)
Affinity DataIC50:  13nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198361(CHEMBL227699 | N-(2,6-dimethylphenyl)-5-[4-(2-pyrr...)
Affinity DataIC50:  15nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198378(CHEMBL389031 | N-(2,6-dimethylphenyl)-5-(4-methoxy...)
Affinity DataIC50:  15nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198377(CHEMBL389422 | N-(2,6-dimethylphenyl)-5-[3-(1-meth...)
Affinity DataIC50:  19nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198365(CHEMBL226613 | N-[5-(4-dimethylaminophenyl)imidazo...)
Affinity DataIC50:  19nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198353(CHEMBL227753 | CHEMBL534948 | N-(2,6-dimethylpheny...)
Affinity DataIC50:  20nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198353(CHEMBL227753 | CHEMBL534948 | N-(2,6-dimethylpheny...)
Affinity DataIC50:  20nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198354(CHEMBL389451 | N-[5-(3,4-dimethoxyphenyl)imidazo[1...)
Affinity DataIC50:  23nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198379(CHEMBL227836 | N-(2,6-dimethylphenyl)-5-[4-(2-morp...)
Affinity DataIC50:  37nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198369(CHEMBL388859 | N-(5-phenylimidazo[1,5-a]pyrazin-8-...)
Affinity DataIC50:  38nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198366(CHEMBL223912 | N-(2,6-dichlorophenyl)-5-phenylimid...)
Affinity DataIC50:  42nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198357(CHEMBL228091 | N-(2,6-dimethylphenyl)-5-(4-fluorop...)
Affinity DataIC50:  42nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198374(4-[8-(2,6-dimethylphenylamino)imidazo[1,5-a]-pyraz...)
Affinity DataIC50:  52nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198358(CHEMBL227652 | N-(2,6-dimethylphenyl)-5-[5-(4-meth...)
Affinity DataIC50:  52nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198376(CHEMBL534947 | N-(2,6-dimethylphenyl)-5-[3-(2-pyrr...)
Affinity DataIC50:  55nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198380(CHEMBL226773 | N-(2-chloro-6-methylphenyl)-6-(3-me...)
Affinity DataIC50:  59nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50151366((2-Chloro-6-methyl-phenyl)-[8-((S)-3-methyl-pipera...)
Affinity DataIC50:  96nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198355(CHEMBL376555 | N-(2,6-dimethylphenyl)-5-pyridin-4-...)
Affinity DataIC50:  108nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198363(CHEMBL224691 | N-(2-chloro-6-methylphenyl)-6-(4-fl...)
Affinity DataIC50:  145nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198381(CHEMBL388820 | N-(2,6-dimethylphenyl)-5-(4-trifluo...)
Affinity DataIC50:  235nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198375(4-[8-(2,6-dimethylphenylamino)imidazo[1,5-a]pyrazi...)
Affinity DataIC50:  235nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198356(4-[8-(2,6-dimethylphenylamino)imidazo[1,5-a]-pyraz...)
Affinity DataIC50:  235nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198367(CHEMBL227859 | N-[5-(4-methoxyphenyl)imidazo[1,5-a...)
Affinity DataIC50:  260nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370960(CHEMBL541412)
Affinity DataIC50:  305nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198362(CHEMBL388136 | N-(2,6-difluorophenyl)-5-phenylimid...)
Affinity DataIC50:  490nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198353(CHEMBL227753 | CHEMBL534948 | N-(2,6-dimethylpheny...)
Affinity DataIC50:  530nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198364(CHEMBL390367 | N-(2-methoxy-6-methylphenyl)-5-phen...)
Affinity DataIC50:  693nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198379(CHEMBL227836 | N-(2,6-dimethylphenyl)-5-[4-(2-morp...)
Affinity DataIC50:  700nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198377(CHEMBL389422 | N-(2,6-dimethylphenyl)-5-[3-(1-meth...)
Affinity DataIC50:  740nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198358(CHEMBL227652 | N-(2,6-dimethylphenyl)-5-[5-(4-meth...)
Affinity DataIC50:  820nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198361(CHEMBL227699 | N-(2,6-dimethylphenyl)-5-[4-(2-pyrr...)
Affinity DataIC50:  950nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198376(CHEMBL534947 | N-(2,6-dimethylphenyl)-5-[3-(2-pyrr...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370960(CHEMBL541412)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198353(CHEMBL227753 | CHEMBL534948 | N-(2,6-dimethylpheny...)
Affinity DataIC50:  2.73E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198382(CHEMBL227376 | N-(2,6-dimethylphenyl)imidazo[1,5-a...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198384(CHEMBL390957 | N-[5-(4-methoxyphenyl)imidazo[1,5-a...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198371(CHEMBL426903 | N-Phenyl-5-phenylimidazo[1,5-a]pyra...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198353(CHEMBL227753 | CHEMBL534948 | N-(2,6-dimethylpheny...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PKCbeta2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198353(CHEMBL227753 | CHEMBL534948 | N-(2,6-dimethylpheny...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198353(CHEMBL227753 | CHEMBL534948 | N-(2,6-dimethylpheny...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Zap70More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198353(CHEMBL227753 | CHEMBL534948 | N-(2,6-dimethylpheny...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SykMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50198359(CHEMBL388807 | N-methyl-N-phenyl-5-phenylimidazo[1...)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed