TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 108nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 145nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 235nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 235nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 235nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 305nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 693nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of cSrc in COS7 cells by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PKCbeta2More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Zap70More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SykMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of cSrc by coupled spectrophotometric enzyme assayMore data for this Ligand-Target Pair