Affinity DataKi: 1nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET-based competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to PPARgamma (unknown origin) assessed as inhibition constant by Lanthascreen TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 142nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 151nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 195nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity to PPARgamma (unknown origin) assessed as inhibition constant by Lanthascreen TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 267nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 272nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 276nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 284nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET-based competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 354nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET-based competitive binding assayMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 417nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 431nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 449nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Binding affinity to PPARgamma (unknown origin) by TR-FRET-based competitive binding assayMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
Affinity DataKi: 590nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 612nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 662nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 810nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 818nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 867nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 1.07E+3nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+3nMAssay Description:Partial agonist activity at PPARgamma (unknown origin) by TR-FRET-based competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.13E+3nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+3nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity to PPARgamma (unknown origin) assessed as inhibition constant by Lanthascreen TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 1.88E+3nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 2.05E+3nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
Affinity DataKi: 2.19E+3nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 3.01E+3nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of human BACE1More data for this Ligand-Target Pair