Affinity DataKi: 0.130nMAssay Description:Binding affinity to 5HT2A receptorMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity for rat GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:Binding affinity to 5HT2A receptorMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity for rat GABA-A receptor alpha-3-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]MDL from rat 5HT2A receptor expressed in GF62 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity for rat GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-1-(arg)-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]MDL from rat 5HT2A receptor expressed in GF62 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr,gly,val)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity for rat GABA-A receptor alpha-3-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity for rat GABA-A receptor alpha-3-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr,gly)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr,gly)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr,gly)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]MDL from rat 5HT2A receptor expressed in GF62 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity for rat GABA-A receptor alpha-6-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr,gly,val)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr,gly)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity for rat GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity for rat GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his)-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity for rat GABA-A receptor alpha-3-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
UniversitÄT Heidelberg
Curated by PDSP Ki Database
UniversitÄT Heidelberg
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Binding affinity for rat GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr,gly,val)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his)-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Binding affinity for rat GABA-A receptor alpha-6-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(RAT)
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his)-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Heidelberg
Curated by ChEMBL
Heidelberg
Curated by ChEMBL
Affinity DataKi: 106nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-1-(arg)-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair