Affinity DataKi: 0.115nMAssay Description:Displacement of CA200645 from NLuc human A3 receptor expressed in HEK293 cells assessed as inhibition constant by NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.115nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.589nMAssay Description:Displacement of CA200645 from NLuc human A1 receptor expressed in HEK293 cells assessed as inhibition constant by NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity to wild type A1R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor T257 6.58A mutant expressed in HEK293 cells measured at 10 mins by NanoBR...More data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of CA200645 from NLuc human A1 receptor expressed in HEK293 cells assessed as inhibition constant by NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to wild type A1R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of CA200645 from NLuc human A3 receptor expressed in HEK293 cells assessed as inhibition constant by NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity to wild type human A1R in presence of CA200645 by saturation NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to wild type A1R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity to human A1R H251 6.52A mutant in presence of CA200645 by saturation NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity to human A1R L250 6.51A mutant in presence of CA200645 by saturation NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bi...More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bi...More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bi...More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity to human A1R E172 5.30A mutant in presence of CA200645 by saturation NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bi...More data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Displacement of CA200645 from NLuc human A1 receptor expressed in HEK293 cells assessed as inhibition constant by NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity to wild type A1R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bi...More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity to wild type A1R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Inhibition of CA200645 binding to wild type NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured at 10 mins by NanoBRET compe...More data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bi...More data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bi...More data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Binding affinity to wild type A1R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Displacement of CA200645 from NLuc human A3 receptor expressed in HEK293 cells assessed as inhibition constant by NanoBRET binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bi...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor N70 2.65A mutant expressed in HEK293 cells measured at 10 mins by NanoBRE...More data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Displacement of [3H]CPX from human Adenosine A1 receptor expressed in DDT1MF-2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor T257 6.58A mutant expressed in HEK293 cells measured at 10 mins by NanoBR...More data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Binding affinity to wild type A3R (unknown origin) expressed in CHO-K1 cells assessed as equilibrium binding affinity constant by nanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused human adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bi...More data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells measured for 10 mins by NanoBRET competition bind...More data for this Ligand-Target Pair