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Found 192 with Last Name = 'lalka' and Initial = 'gk'
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50058855((S)-2-Butoxycarbonylamino-3-{2-[(R)-3-(4-carbamimi...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of [125I]fibrinogen binding to purified platelet Fibrinogen ReceptorMore data for this Ligand-Target Pair
LigandPNGBDBM50031491(2-propyl-4-(methythio)-1-[[[2'-[(propylamino)carbo...)
Affinity DataIC50:  0.300nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283002(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50:  0.600nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283000(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283182(3-[3-Fluoro-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50:  0.900nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50032364(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50032362(3-(2'-Isopentyloxycarbonylsulfamoyl-3-fluoro-biphe...)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50032362(3-(2'-Isopentyloxycarbonylsulfamoyl-3-fluoro-biphe...)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283005(3-(2'-Butyloxycarbonylsulfamoyl-3-bromo-biphenyl-4...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283169(2-Propyl-5-(4-pyridin-2-yl-piperazin-1-ylmethyl)-3...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM36645(CHEMBL291582 | L-707,581)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283008(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283006(3-(2'-Butyloxycarbonylsulfamoyl-biphenyl-4-ylmethy...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283001(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283003(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283000(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283159(5-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-2-pr...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283161(2-Propyl-5-(4-pyridin-2-yl-piperazine-1-carbonyl)-...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283162(5-[(Butyl-butyryl-amino)-methyl]-3-(2'-butyrylsulf...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283176(5-(1-Benzyl-3-phenyl-ureidomethyl)-2-propyl-3-[2'-...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283174(5-Dipentylaminomethyl-2-propyl-3-[2'-(1H-tetrazol-...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283179(5-((R)-2-Methyl-4-phenyl-piperazin-1-ylmethyl)-2-p...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283183(2-Propyl-5-(4-pyrimidin-2-yl-piperazin-1-ylmethyl)...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283185(5-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-2-pro...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283188(5-(4-Phenyl-piperidin-1-ylmethyl)-2-propyl-3-[2'-(...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283164(2-Butyl-5-(4-pyridin-2-yl-piperazin-1-ylmethyl)-3-...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50049179(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM82428(CAS_124750-95-4 | CB91356279 | CHEMBL443269 | DuP ...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283009(4'-(4-Ethyl-5-formyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283007(3-(2'-Butyloxycarbonylsulfamoyl-3-methyl-biphenyl-...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283178(5-[(Benzyl-butyl-amino)-methyl]-2-propyl-3-[2'-(1H...)
Affinity DataIC50:  3nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50032351(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50032364(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283165(5-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-2-pro...)
Affinity DataIC50:  3nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50049196(3-[3-Bromo-2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50283002(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50049178(2-Propyl-5-(4-pyridin-2-yl-piperazin-1-ylmethyl)-3...)
Affinity DataIC50:  4.20nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283171(5-(4-Phenyl-piperazin-1-ylmethyl)-2-propyl-3-[2'-(...)
Affinity DataIC50:  5nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283175(5-(4-Benzoyl-piperazin-1-ylmethyl)-2-propyl-3-[2'-...)
Affinity DataIC50:  5nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50406795(Cozaar | LOSARTAN POTASSIUM)
Affinity DataIC50:  5.5nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50282999(4'-(5-Acetyl-4-ethyl-2-propyl-imidazol-1-ylmethyl)...)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283170(1-[4-(2-pentanyloxycarbonylsulfamoylphenyl)benzyl]...)
Affinity DataIC50:  6nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283181(5-(tert-Butoxycarbonylamino-methyl)-2-propyl-3-[2'...)
Affinity DataIC50:  6nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283160(3-(2'-Hexanoylsulfamoyl-biphenyl-4-ylmethyl)-2-pro...)
Affinity DataIC50:  6nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283173(3-(2'-Benzoylsulfamoyl-biphenyl-4-ylmethyl)-2-prop...)
Affinity DataIC50:  6nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283012(3-(2'-Butyloxycarbonylsulfamoyl-3-nitro-biphenyl-4...)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50032351(3-(2'-Butyloxycarbonylsulfamoyl-3-chloro-biphenyl-...)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT2 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50283004(5-Ethyl-3-[3-fluoro-2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  7nMAssay Description:Displacement of [125I]- Ang II from angiotensin II AT1 receptor in rat adrenal cortical microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283190(4-benzyl(phenyl)carboxamidomethyl-1-{4-[2-(isobuty...)
Affinity DataIC50:  8nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283186(5-[(Benzyl-tert-butoxycarbonyl-amino)-methyl]-2-pr...)
Affinity DataIC50:  9nMAssay Description:In vitro binding affinity of compound against Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails Article
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