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Found 74 with Last Name = 'larsson' and Initial = 'lg'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85827((R)-3-[Isopropyl(propyl)amino]-3,4-dihydro-2H-1-be...)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  0.590nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85826((R)-N-Isopropyl-3-[isopropyl(propyl)amino]-3,4-dih...)
Affinity DataKi:  4.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  45nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi:  47nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369357(CHEMBL1201939)
Affinity DataKi:  60nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  67nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  79nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM85827((R)-3-[Isopropyl(propyl)amino]-3,4-dihydro-2H-1-be...)
Affinity DataKi:  88nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM85826((R)-N-Isopropyl-3-[isopropyl(propyl)amino]-3,4-dih...)
Affinity DataKi:  240nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064466(CHEMBL58961 | Morpholin-4-yl-[8-(morpholin-2-ylmet...)
Affinity DataKi:  240nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064462(8-(Morpholin-2-ylmethoxy)-2H-chromene-3-carbonitri...)
Affinity DataKi:  250nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369355(CHEMBL1202783)
Affinity DataKi:  275nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  340nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064464(5-(Morpholin-2-ylmethoxy)-3,4-dihydro-naphthalene-...)
Affinity DataKi:  445nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM85826((R)-N-Isopropyl-3-[isopropyl(propyl)amino]-3,4-dih...)
Affinity DataKi:  500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM85827((R)-3-[Isopropyl(propyl)amino]-3,4-dihydro-2H-1-be...)
Affinity DataKi:  500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM85826((R)-N-Isopropyl-3-[isopropyl(propyl)amino]-3,4-dih...)
Affinity DataKi:  500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM85827((R)-3-[Isopropyl(propyl)amino]-3,4-dihydro-2H-1-be...)
Affinity DataKi:  500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(1A) dopamine receptor(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM85827((R)-3-[Isopropyl(propyl)amino]-3,4-dihydro-2H-1-be...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor using [3H]QNB as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(1A) dopamine receptor(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(BOVINE)
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM85826((R)-N-Isopropyl-3-[isopropyl(propyl)amino]-3,4-dih...)
Affinity DataKi:  1.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064467(8-(Piperidin-3-ylmethoxy)-2H-chromene-3-carbonitri...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  1.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalanin peptides(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  2.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalanin peptides(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  2.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 6(RAT)
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >3.00E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 6 receptor from CHO cell membranes using [3H]5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064465(8-(4-Methyl-morpholin-2-ylmethoxy)-2H-chromene-3-c...)
Affinity DataKi:  3.60E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astrazeneca R&D

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 6(RAT)
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor 3(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor 3(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Preclinical R & D, Astra Arcus

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
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