Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 8.80nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT2 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 408nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 1.35E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta scintillation counting analys...More data for this Ligand-Target Pair
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [125I]Sar-Ile-angiotensin 2 from human AT1 receptor expressed in HEK293 cells incubated for 240 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using bufuralol as substrate preincubated for 3 mins followed by NADPH addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP2C9 in human liver microsomes using diclofenac as substrate preincubated for 3 mins followed by NADPH addition by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomes using diclofenac as substrate preincubated for 3 mins followed by NADPH addition by LC-MS/MS analysisMore data for this Ligand-Target Pair