Affinity DataKi: 0.140nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
New York University
Curated by ChEMBL
New York University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]-haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
New York University
Curated by ChEMBL
New York University
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]- haloperidolMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
New York University
Curated by ChEMBL
New York University
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]- haloperidolMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 18.3nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 18.3nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 19.4nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 19.4nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 24.7nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 24.7nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 26.4nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 26.4nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 80nM ΔG°: -40.1kJ/molepH: 7.4 T: 2°CAssay Description:Affinities for D3-dopaminergic, D2-dopaminergic and beta2-adrenergic receptors were determined by radioligand competition binding at the National Ins...More data for this Ligand-Target Pair
Affinity DataKi: 100nM ΔG°: -39.6kJ/molepH: 7.4 T: 2°CAssay Description:Affinities for D3-dopaminergic, D2-dopaminergic and beta2-adrenergic receptors were determined by radioligand competition binding at the National Ins...More data for this Ligand-Target Pair
Affinity DataKi: 100nM ΔG°: -39.6kJ/molepH: 7.4 T: 2°CAssay Description:Affinities for D3-dopaminergic, D2-dopaminergic and beta2-adrenergic receptors were determined by radioligand competition binding at the National Ins...More data for this Ligand-Target Pair
Affinity DataKi: 100nM ΔG°: -39.6kJ/molepH: 7.4 T: 2°CAssay Description:Affinities for D3-dopaminergic, D2-dopaminergic and beta2-adrenergic receptors were determined by radioligand competition binding at the National Ins...More data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Inhibitory activity against thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 200nM ΔG°: -37.9kJ/molepH: 7.4 T: 2°CAssay Description:Affinities for D3-dopaminergic, D2-dopaminergic and beta2-adrenergic receptors were determined by radioligand competition binding at the National Ins...More data for this Ligand-Target Pair
Affinity DataKi: 200nM ΔG°: -37.9kJ/molepH: 7.4 T: 2°CAssay Description:Affinities for D3-dopaminergic, D2-dopaminergic and beta2-adrenergic receptors were determined by radioligand competition binding at the National Ins...More data for this Ligand-Target Pair
Affinity DataKi: 200nM ΔG°: -37.9kJ/molepH: 7.4 T: 2°CAssay Description:Affinities for D3-dopaminergic, D2-dopaminergic and beta2-adrenergic receptors were determined by radioligand competition binding at the National Ins...More data for this Ligand-Target Pair
Affinity DataKi: 200nM ΔG°: -37.9kJ/molepH: 7.4 T: 2°CAssay Description:Affinities for D3-dopaminergic, D2-dopaminergic and beta2-adrenergic receptors were determined by radioligand competition binding at the National Ins...More data for this Ligand-Target Pair
Affinity DataKi: 200nM ΔG°: -37.9kJ/molepH: 7.4 T: 2°CAssay Description:Affinities for D3-dopaminergic, D2-dopaminergic and beta2-adrenergic receptors were determined by radioligand competition binding at the National Ins...More data for this Ligand-Target Pair