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Found 43 with Last Name = 'lescrinier' and Initial = 'e'
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50544145(CHEMBL4636583)
Affinity DataKi:  88nMAssay Description:Inhibition of Escherichia coli BL21(DE3) ileRS overexpressed in Escherichia coli Rosetta2(DE3) assessed as reduction in tRNA aminoacylation preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoleucine--tRNA ligase(Escherichia coli)
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50544146(CHEMBL4648043)
Affinity DataKi:  114nMAssay Description:Inhibition of Escherichia coli BL21(DE3) ileRS overexpressed in Escherichia coli Rosetta2(DE3) assessed as reduction in tRNA aminoacylation preincuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351763(CHEMBL1823492)
Affinity DataIC50:  290nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351763(CHEMBL1823492)
Affinity DataIC50:  570nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351764(CHEMBL1823500)
Affinity DataIC50:  910nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351765(CHEMBL1823505)
Affinity DataIC50:  4.84E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351771(CHEMBL1823504)
Affinity DataIC50:  6.93E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351758(CHEMBL1823503)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351759(CHEMBL1823493)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351760(CHEMBL1823498)
Affinity DataIC50:  8.03E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351761(CHEMBL1823501)
Affinity DataIC50:  8.61E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351762(CHEMBL1823494)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351766(CHEMBL1823502)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351767(CHEMBL1823496)
Affinity DataIC50:  2.78E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351759(CHEMBL1823493)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351770(CHEMBL1823499)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351768(CHEMBL1823495)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351767(CHEMBL1823496)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351769(CHEMBL1823497)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351760(CHEMBL1823498)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351770(CHEMBL1823499)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351764(CHEMBL1823500)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351761(CHEMBL1823501)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351766(CHEMBL1823502)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351758(CHEMBL1823503)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351771(CHEMBL1823504)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351765(CHEMBL1823505)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351769(CHEMBL1823497)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase ThyA(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351762(CHEMBL1823494)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis His-tagged ThyA-mediated dTMP synthesis expressed in BL21 (DE3) Escherichia coli RbCl cells after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFlavin-dependent thymidylate synthase(Mycobacterium tuberculosis)
Katholieke Universiteit Leuven

Curated by ChEMBL
LigandPNGBDBM50351768(CHEMBL1823495)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ThyX-mediated dTMP synthesis using [5-3H]dUMP as substrate after 10 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507722(CHEMBL4517342)
Affinity DataKd: >3.00E+4nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507723(CHEMBL4461988)
Affinity DataKd: >3.00E+4nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507724(CHEMBL4529993)
Affinity DataKd:  400nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507725(CHEMBL4576567)
Affinity DataKd:  770nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50086260(CHEMBL3425846)
Affinity DataKd:  52nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507726(CHEMBL4522263)
Affinity DataKd:  7.60E+3nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507720(CHEMBL4463819)
Affinity DataKd: >3.00E+4nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507728(CHEMBL4451350)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507729(CHEMBL4574041)
Affinity DataKd:  520nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507730(CHEMBL4579614)
Affinity DataKd:  860nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507731(CHEMBL4558505)
Affinity DataKd:  41nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507721(CHEMBL4454241)
Affinity DataKd:  3.20E+3nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50507727(CHEMBL4525511)
Affinity DataKd:  3.20E+3nMAssay Description:Binding affinity to wild type DNA-tagged human GAK (G13 to Y338 residues) expressed in bacterial expression system by quantitative PCR based KINOMEsc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed