TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 0.116nMAssay Description:Displacement of [3H]cytisine from rat alpha4beta2 nAChR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 0.165nMAssay Description:Displacement of [3H]cytisine from rat alpha4beta2 nAChR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 0.208nMAssay Description:Displacement of [3H]cytisine from rat alpha4beta2 nAChR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [3H]cytisine from rat alpha4beta2 nAChR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]cytisine from rat alpha4beta2 nAChR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 1.06nMAssay Description:Displacement of [3H]cytisine from rat alpha4beta2 nAChR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 6.53nMAssay Description:Displacement of [3H]cytisine from rat alpha4beta2 nAChR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Displacement of [125I]alphaBungarotoxin from alpha7 nAchR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 401nMAssay Description:Displacement of [125I]alphaBungarotoxin from alpha7 nAchR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [125I]alphaBungarotoxin from alpha7 nAchR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [125I]alphaBungarotoxin from alpha7 nAchR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [125I]alphaBungarotoxin from alpha7 nAchR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Ensicaen-Université
Curated by ChEMBL
Ensicaen-Université
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [125I]alphaBungarotoxin from alpha7 nAchR in rat brain cell membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Servier, Chemistry Research Division A
Curated by PDSP Ki Database
Affinity DataEC50: 4.17E+3nMAssay Description:Positive allosteric modulation of GluA2 receptor in rat embryonic cortex neuron assessed as increase of AMPA-induced membrane depolarization by fluor...More data for this Ligand-Target Pair
Affinity DataEC50: 3.13E+3nMAssay Description:Positive allosteric modulation of GluA2 receptor in rat embryonic cortex neuron assessed as increase of AMPA-induced membrane depolarization by fluor...More data for this Ligand-Target Pair
Affinity DataEC50: 2.50E+3nMAssay Description:Positive allosteric modulation of GluA2 receptor in rat embryonic cortex neuron assessed as increase of AMPA-induced membrane depolarization by fluor...More data for this Ligand-Target Pair
Affinity DataEC50: 900nMAssay Description:Positive allosteric modulation of GluA2 receptor in rat embryonic cortex neuron assessed as increase of AMPA-induced membrane depolarization by fluor...More data for this Ligand-Target Pair
Affinity DataEC50: 2.25E+4nMAssay Description:Positive allosteric modulation of GluA2 receptor in rat embryonic cortex neuron assessed as increase of AMPA-induced membrane depolarization by FLIPR...More data for this Ligand-Target Pair
Affinity DataEC50: 4.83E+3nMAssay Description:Positive allosteric modulation of GluA2 receptor in rat embryonic cortex neuron assessed as increase of AMPA-induced membrane depolarization by fluor...More data for this Ligand-Target Pair
Affinity DataKd: 350nMAssay Description:Binding affinity to GluA2-LBD-L483Y-N754S complex (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 9.80E+3nMAssay Description:Binding affinity to GluA2-LBD-L483Y-N754S complex (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+6nMAssay Description:Binding affinity to GluA2-LBD-L483Y-N754S complex (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 5.60E+3nMAssay Description:Binding affinity to GluA2-LBD-L483Y-N754S complex (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair