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Found 107 with Last Name = 'lesur' and Initial = 'b'
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291029((2R,3R,4R,5S)-2-Hydroxymethyl-1-((E)-3-trimethylsi...)
Affinity DataKi:  0.150nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291029((2R,3R,4R,5S)-2-Hydroxymethyl-1-((E)-3-trimethylsi...)
Affinity DataKi:  2.30nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291026((2R,3R,4R,5S)-1-[(E)-3-(Dimethyl-phenyl-silanyl)-a...)
Affinity DataKi:  3nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291026((2R,3R,4R,5S)-1-[(E)-3-(Dimethyl-phenyl-silanyl)-a...)
Affinity DataKi:  4nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365043(CHEMBL1951055)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291031((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  8nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365051(CHEMBL1951060)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291031((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  8nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365052(CHEMBL1951061)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291023((2R,3R,4R,5S)-1-[(E)-3-(tert-Butyl-dimethyl-silany...)
Affinity DataKi:  10nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365053(CHEMBL1951062)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291020((2R,3R,4R,5S)-1-[3-(Dimethyl-phenyl-silanyl)-propy...)
Affinity DataKi:  10nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365043(CHEMBL1951055)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291021((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  16nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291034((2R,3R,4R,5S)-2-Hydroxymethyl-1-(5-trimethylsilany...)
Affinity DataKi:  16nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291020((2R,3R,4R,5S)-1-[3-(Dimethyl-phenyl-silanyl)-propy...)
Affinity DataKi:  17nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291030((2R,3R,4R,5S)-1-[4-(Dimethyl-phenyl-silanyl)-butyl...)
Affinity DataKi:  18nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365054(CHEMBL1951063)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM18353((2R,3R,4R,5S)-2-(hydroxymethyl)-1-methylpiperidine...)
Affinity DataKi:  20nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  24nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291020((2R,3R,4R,5S)-1-[3-(Dimethyl-phenyl-silanyl)-propy...)
Affinity DataKi:  27nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291027((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  28nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365044(CHEMBL1951052)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291034((2R,3R,4R,5S)-2-Hydroxymethyl-1-(5-trimethylsilany...)
Affinity DataKi:  33nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365052(CHEMBL1951061)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291030((2R,3R,4R,5S)-1-[4-(Dimethyl-phenyl-silanyl)-butyl...)
Affinity DataKi:  39nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291021((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  40nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365043(CHEMBL1951055)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291031((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  50nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291026((2R,3R,4R,5S)-1-[(E)-3-(Dimethyl-phenyl-silanyl)-a...)
Affinity DataKi:  50nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291032((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  55nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365043(CHEMBL1951055)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291027((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  64nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365046(CHEMBL1951054)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291034((2R,3R,4R,5S)-2-Hydroxymethyl-1-(5-trimethylsilany...)
Affinity DataKi:  70nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365053(CHEMBL1951062)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291023((2R,3R,4R,5S)-1-[(E)-3-(tert-Butyl-dimethyl-silany...)
Affinity DataKi:  87nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365047(CHEMBL1951056)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291029((2R,3R,4R,5S)-2-Hydroxymethyl-1-((E)-3-trimethylsi...)
Affinity DataKi:  100nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365051(CHEMBL1951060)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365045(CHEMBL1951053)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291028((2R,3R,4R,5S)-1-(Dimethyl-propyl-silanylmethyl)-2-...)
Affinity DataKi:  110nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291031((2R,3R,4R,5S)-2-Hydroxymethyl-1-(3-trimethylsilany...)
Affinity DataKi:  120nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291021((2R,3R,4R,5S)-2-Hydroxymethyl-1-(4-trimethylsilany...)
Affinity DataKi:  120nMAssay Description:In vitro inhibition constant against rat small intestinal glucoamylaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetLysosomal alpha-glucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  150nMAssay Description:Tested in vitro for the inhibition constant against human lysosomal alpha-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291022((2R,3R,4R,5S)-2-Hydroxymethyl-1-trimethylsilanylme...)
Affinity DataKi:  150nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291033((2R,3R,4R,5S)-1-[(Dimethyl-phenyl-silanyl)-methyl]...)
Affinity DataKi:  160nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365044(CHEMBL1951052)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50291025((2R,3R,4R,5S)-2-Hydroxymethyl-1-((E)-4-trimethylsi...)
Affinity DataKi:  220nMAssay Description:Tested in vitro for the inhibition constant against rat small intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365054(CHEMBL1951063)
Affinity DataKi:  244nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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