BindingDB PrimarySearch

Found 469 with Last Name = 'li' and Initial = 'yy'

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

Ki: 0.380nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562185(CHEMBL4746910)

Ki: 1.30nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562179(CHEMBL4739972)

Ki: 3nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)

Ki: 3.30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed PDB

3D Structure (crystal)

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562176(CHEMBL4778377)

Ki: 5.10nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562184(CHEMBL4744206)

Ki: 13nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562183(CHEMBL4760742)

Ki: 20nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562181(CHEMBL4747537)

Ki: 22nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562180(CHEMBL4796195)

Ki: 34nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)

Ki: 35nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG PC cid PC sid PDB Patents Similars

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562186(CHEMBL4761905)

Ki: 40nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562177(CHEMBL4763056)

Ki: 42nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562179(CHEMBL4739972)

Ki: 160nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562173(CHEMBL4778965)

Ki: 956nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562185(CHEMBL4746910)

Ki: >1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562186(CHEMBL4761905)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562187(CHEMBL4765186)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562178(CHEMBL4740343)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562184(CHEMBL4744206)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562183(CHEMBL4760742)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562180(CHEMBL4796195)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562181(CHEMBL4747537)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562182(CHEMBL4744466)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562187(CHEMBL4765186)

Ki: >1.00E+3nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562174(CHEMBL4759158)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562178(CHEMBL4740343)

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562177(CHEMBL4763056)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562176(CHEMBL4778377)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562175(CHEMBL4749663)

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562175(CHEMBL4749663)

Ki: 3.18E+3nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Guangdong Medical University

Curated by ChEMBL

BDBM50562173(CHEMBL4778965)

Ki: 3.19E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

PDB
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Sigma intracellular receptor 2(Rattus norvegicus (Rat))
Guangdong Medical University

Curated by ChEMBL

BDBM50562174(CHEMBL4759158)

Ki: 1.15E+4nMAssay Description:Displacement of [125I]-RHM-4 from sigma 2 receptor in rat liver membranes after 120 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

PC cid PC sid

Details Article PubMed

Mitogen-activated protein kinase 10(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL

BDBM50495031(CHEMBL3099975)

IC50: 1nMAssay Description:Inhibition of JNK3 (39 to 402 amino acids) (unknown origin) expressed in Escherichia coli BL21(DE3) using biotinylated ATF2 as substrate after 15 min...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Vitamin D3 receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)

IC50: 1.40nMAssay Description:Displacement of fluormone VDR red from human full-length VDR after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
KEGG MMDB PC cid PC sid PDB Patents Similars

Details Article PubMed DrugBank

Xanthine dehydrogenase/oxidase(Homo sapiens (Human))
Soochow University

Curated by ChEMBL

BDBM50140241(Allopurinol | Aloral | Aluline 100 | Aluline 300 |...)

IC50: 3.60nMAssay Description:Inhibition of xanthine oxidase (unknown origin) assessed as reduction in uric acid formation preincubated for 5 mins followed by addition of xanthine...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase MCE
PC cid PC sid Similars

Details Article PubMed

Mitogen-activated protein kinase 14(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL

BDBM50563622(CHEMBL4778963)

IC50: 4nMAssay Description:Inhibition of recombinant human p38alpha expressed in Escherichia coli assessed as incoporation of [33]Pi after 60 mins in presence of [gamma-33P]-AT...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Mitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL

BDBM50495026(CHEMBL3099962)

IC50: 4nMAssay Description:Inhibition of p38 (unknown origin)More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

TGF-beta receptor type-1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL

BDBM50563622(CHEMBL4778963)

IC50: 4nMAssay Description:Inhibition of recombinant human GST-fused ALK5 expressed in baculovirus infected Sf9 cells assessed as incoporation of [33]Pi after 60 mins in presen...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Mitogen-activated protein kinase 10(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL

BDBM50340629(8-methoxy-7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-mor...)

IC50: 4nMAssay Description:Inhibition of JNK3 by HRTFMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Mitogen-activated protein kinase 10(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL

BDBM50303639(CHEMBL571626 | N-(4-(2-(4-(1H-1,2,3-Triazol-1-yl)p...)

IC50: 4nMAssay Description:Inhibition of JNK3 by time resolved fluorescence assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid

Details Article PubMed

TGF-beta receptor type-1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL

BDBM50563621(CHEMBL4748823)

PDB MMDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

TGF-beta receptor type-1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL

BDBM50563624(CHEMBL4747557)

IC50: 5nMAssay Description:Inhibition of recombinant human GST-fused ALK5 expressed in baculovirus infected Sf9 cells assessed as incoporation of [33]Pi after 60 mins in presen...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

TGF-beta receptor type-1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL

BDBM50563620(CHEMBL4779584)

PDB MMDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Xanthine dehydrogenase/oxidase(Homo sapiens (Human))
Soochow University

Curated by ChEMBL

BDBM50424969(CHEMBL2316146 | US9409845, Table 1, Compound 7: (2...)

IC50: 5.70nMAssay Description:Inhibition of xanthine oxidase (unknown origin) assessed as reduction in uric acid formation preincubated for 5 mins followed by addition of xanthine...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

TGF-beta receptor type-1(Homo sapiens (Human))
Yanbian University

Curated by ChEMBL

BDBM50563623(CHEMBL4780141)

IC50: 6nMAssay Description:Inhibition of recombinant human GST-fused ALK5 expressed in baculovirus infected Sf9 cells assessed as incoporation of [33]Pi after 60 mins in presen...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Mitogen-activated protein kinase 10(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL

BDBM50342502(CHEMBL1771718 | N-(4-(3,5-dimethyl-1H-1,2,4-triazo...)

IC50: 7nMAssay Description:Inhibition of JNK3 assessed as formation of phospho-Thr71-ATF-2 from biotinylated-ATF2 by HTRF assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Mitogen-activated protein kinase 10(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL

BDBM50303638(4-(4-(4-(Methylsulfonamido)phenyl)pyrimidin-2-ylam...)

IC50: 7nMAssay Description:Inhibition of JNK3 by time resolved fluorescence assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid Similars

Details Article PubMed

Mitogen-activated protein kinase 10(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL

BDBM92524(Aminopyrazole inhibitor, 3576)

IC50: 7nMpH: 7.0 T: 2°CAssay Description:Homogeneous time-resolved fluorescence assay is an enzyme inhibition studies that were performed in 384-well polystyrene homogeneous time-resolved fl...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase PC cid PC sid Similars

Details Article PubMed

Mitogen-activated protein kinase 10(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL

BDBM50495026(CHEMBL3099962)

IC50: 7nMAssay Description:Inhibition of JNK3 (39 to 402 amino acids) (unknown origin) expressed in Escherichia coli BL21(DE3) using biotinylated ATF2 as substrate after 15 min...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Mitogen-activated protein kinase 10(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL

BDBM50340611(CHEMBL1761566 | N-(4-(3-morpholino-1H-1,2,4-triazo...)

IC50: 7nMAssay Description:Inhibition of JNK3 by HRTFMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid

Details Article PubMed

Displayed 1 to 50 (of 469 total ) | Next | Last >>

Filter my 469 hits

Targets 19▿
- Mitogen-activated protein kinase 10 129
- Mitogen-activated protein kinase 8 77
- Isoform Alpha-1 of Mitogen-activated protein kinase 10 (Alpha-1) 9-402] 46
- Histone deacetylase 8 31
- 72 kDa type IV collagenase 31
- Transcription factor Jun 22
- Mitogen-activated protein kinase 11/12/13/14 18
- TGF-beta receptor type-1 16
- Sigma intracellular receptor 2 16
- Sigma non-opioid intracellular receptor 1 16
- Mitogen-activated protein kinase 14 16
- 5'-AMP-activated protein kinase catalytic subunit alpha-2/subunit beta-1/subunit gamma-1 15
- Xanthine dehydrogenase/oxidase 10
- Mitogen-activated protein kinase 13 8
- Vitamin D3 receptor 8
- Retinoic acid receptor RXR-alpha/Vitamin D3 receptor 4
- 5'-AMP-activated protein kinase catalytic subunit alpha-1 3
- Reverse transcriptase 2
- 5'-AMP-activated protein kinase catalytic subunit alpha-2 1
- ...
Publications 14▿
- Bioorg Med Chem Lett 19: 3344-7 (2009) 88
- Bioorg Med Chem 20: 5738-44 (2012) 62
- Bioorg Med Chem Lett 21: 1719-23 (2011) 62
- Bioorg Med Chem Lett 24: 161-4 (2014) 46
- Eur J Med Chem 216: (2021) 32
- Eur J Med Chem 209: (2021) 32
- Bioorg Med Chem Lett 21: 2732-5 (2011) 30
- Bioorg Med Chem Lett 17: 6378-82 (2007) 26
- J Biol Chem 284: 12853-61 (2009) 24
- J Med Chem 53: 419-31 (2010) 24
- ACS Med Chem Lett 4: 475-80 (2013) 19
- Eur J Med Chem 157: 1174-1191 (2018) 12
- Bioorg Med Chem 25: 166-174 (2017) 10
- J Nat Prod 59: 1061-5 (1996) 2
Institutions 10▿
- The Scripps Research Institute 250
- Tianjin Medical University 62
- Yanbian University 32
- Guangdong Medical University 32
- Scripps Florida 26
- Translational Research Institute 24
- Chinese Academy Of Sciences 19
- China Pharmaceutical University 12
- Soochow University 10
- National Taiwan University 2
Affinity: 0.38 to 1.0E+6 nM▿
- Ki 32
- IC50 414
- EC50 23
- Affinity ≤ nM
Xtal structures: 6
Docked structures: 1
Catalog Cmpds: 17