BindingDB PrimarySearch

Found 394 with Last Name = 'lin' and Initial = 'js'

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

Ki: 0.280nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580523(CHEMBL5093850)

Ki: 0.310nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580512(CHEMBL5072724)

Ki: 0.490nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580514(CHEMBL5093935)

Ki: 0.600nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50202986(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-ethoxy)-phenyl]...)

Ki: 0.880nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase CHEMBL MCE
PC cid PC sid Patents Similars

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580516(CHEMBL5094415)

Ki: 2.30nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580522(CHEMBL5082650)

Ki: 4nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580517(CHEMBL5084903)

Ki: 4.5nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580517(CHEMBL5084903)

Ki: 4.90nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580520(CHEMBL5082920)

Ki: 6.20nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580515(CHEMBL5088622)

Ki: 7.30nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50316887(2-amino-8-(2-morpholinoethoxy)-4-phenyl-5H-indeno[...)

Ki: 7.5nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580515(CHEMBL5088622)

Ki: 11nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50458224(CHEMBL2297871)

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase PC cid PC sid

Details Article PubMed

Adenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580522(CHEMBL5082650)

Ki: 11nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580513(CHEMBL5094263)

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580515(CHEMBL5088622)

Ki: 12nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580520(CHEMBL5082920)

Ki: 13nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580520(CHEMBL5082920)

Ki: 17nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580517(CHEMBL5084903)

Ki: 19nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580519(CHEMBL5081556)

Ki: 31nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580521(CHEMBL5087059)

Ki: 36nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580518(CHEMBL5089580)

Ki: 36nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580515(CHEMBL5088622)

Ki: 37nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580522(CHEMBL5082650)

Ki: 44nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580520(CHEMBL5082920)

Ki: 48nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580522(CHEMBL5082650)

Ki: 52nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580517(CHEMBL5084903)

Ki: 58nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580519(CHEMBL5081556)

Ki: 104nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580521(CHEMBL5087059)

Ki: 114nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580519(CHEMBL5081556)

Ki: 129nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580518(CHEMBL5089580)

Ki: 133nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580521(CHEMBL5087059)

Ki: 142nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580522(CHEMBL5082650)

Ki: 150nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580515(CHEMBL5088622)

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580519(CHEMBL5081556)

Ki: 180nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580520(CHEMBL5082920)

Ki: 199nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580523(CHEMBL5093850)

Ki: 203nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Histamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50458225(Ciproxifan)

Ki: 224nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase MCE
PC cid PC sid

Details Article PubMed

Adenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580517(CHEMBL5084903)

Ki: 231nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

D(3) dopamine receptor(Homo sapiens)
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580515(CHEMBL5088622)

Ki: 290nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50202986(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-ethoxy)-phenyl]...)

Ki: 295nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase CHEMBL MCE
PC cid PC sid Patents Similars

Details Article PubMed

Adenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580518(CHEMBL5089580)

Ki: 331nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

D(3) dopamine receptor(Homo sapiens)
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580522(CHEMBL5082650)

Ki: 364nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580521(CHEMBL5087059)

Ki: 367nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50316887(2-amino-8-(2-morpholinoethoxy)-4-phenyl-5H-indeno[...)

Ki: 430nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Purchase CHEMBL PC cid PC sid Patents Similars

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580512(CHEMBL5072724)

Ki: 717nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580513(CHEMBL5094263)

Ki: 828nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580519(CHEMBL5081556)

Ki: 846nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Adenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf

Curated by ChEMBL

BDBM50580514(CHEMBL5093935)

Ki: 941nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Displayed 1 to 50 (of 394 total ) | Next | Last >>

Filter my 394 hits

Targets 15▿
- RAC-alpha serine/threonine-protein kinase 230
- Short transient receptor potential channel 3 32
- Short transient receptor potential channel 6 32
- Adenosine receptor A3 16
- Adenosine receptor A2b 16
- Adenosine receptor A2a 16
- Adenosine receptor A1 15
- Histamine H3 receptor 14
- Reverse transcriptase/RNaseH 12
- D(3) dopamine receptor 2
- Histamine H1 receptor 2
- D(2) dopamine receptor 2
- D(1B) dopamine receptor 2
- Histamine H4 receptor 2
- Amine oxidase [flavin-containing] B 1
- ...
Publications 4▿
- US Patent US8541407 (2013) 230
- J Med Chem 64: 8246-8262 (2021) 88
- US Patent US11274091 (2022) 64
- J Med Chem 41: 10-23 (1998) 12
Institutions 4▿
- Arqule 230
- Heinrich Heine University Duesseldorf 88
- Dizal (Jiangsu) Pharmaceutical 64
- Wayne State University School Of Medicine 12
Affinity: 0.28 to 1.0E+5 nM▿
- Ki 85
- IC50 307
- EC50 2
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 6