TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Binding affinity at Mutant (H272E) human adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 0.540nMAssay Description:Binding affinity at wild-type Adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.730nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.770nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 0.870nMAssay Description:Binding affinity at wild-type Adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.940nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the presence of GTPMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity at wild-type Adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.46nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity at wild-type Adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Binding affinity at Mutant (H272E) human adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.13nMAssay Description:Binding affinity at human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Binding affinity at Mutant (H272E) human adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Binding affinity at rat adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Binding affinity at wild-type Adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Binding affinity at wild-type Adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:GTP-induced shift at rat Adenosine A1 receptor (A1AR)More data for this Ligand-Target Pair
Affinity DataKi: 6.69nMAssay Description:Binding affinity at rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Binding affinity at rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 9.60nMAssay Description:Binding affinity at Mutant (H272E) human adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 9.90nMAssay Description:Binding affinity at Mutant (H272E) human adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity at rat adenosine A3 receptor in RBL-2H3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A2A receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity at rat adenosine A3 receptor in RBL-2H3 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A2A receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A2A receptor in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A2A receptor in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A2A receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A2A receptor in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity at rat adenosine A3 receptor in RBL-2H3 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A2A receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Binding affinity at rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 14.7nMAssay Description:Binding affinity at rat adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the presence of GTPMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 19.6nMAssay Description:Binding affinity at wild-type Adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 20.1nMAssay Description:Binding affinity at Mutant (H272E) human adenosine A3 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity at rat Adenosine A1 receptor in the absence of GTPMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Binding affinity at rat brain Adenosine A2A receptor in CHO cellsMore data for this Ligand-Target Pair