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Found 19 with Last Name = 'lipinski' and Initial = 'pf'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50081529((S)-2-Amino-N-{(R)-1-[({(S)-2-[N'-((S)-2-amino-3-p...)
Affinity DataIC50:  0.740nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [Leu-3,4,5-3H(N)]-Substance P from NK1 receptor in rat brain homogenate measured after 60 mins by microbeta scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50208162(CHEMBL3904919)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50208162(CHEMBL3904919)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [3H]DELT2 from DOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50208161(CHEMBL3932836)
Affinity DataIC50:  4.20nMAssay Description:Displacement of [Leu-3,4,5-3H(N)]-Substance P from NK1 receptor in rat brain homogenate measured after 60 mins by microbeta scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50081523((S)-2-Amino-N-((R)-1-{[((S)-1-hydrazinocarbonyl-2-...)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [3H]DAMGO from MOR in Sprague-Dawley rat brain homogenate measured after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50208161(CHEMBL3932836)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50081529((S)-2-Amino-N-{(R)-1-[({(S)-2-[N'-((S)-2-amino-3-p...)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]DELT2 from DOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50208161(CHEMBL3932836)
Affinity DataIC50:  74nMAssay Description:Displacement of [3H]DELT2 from DOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropilin-1(Rattus norvegicus)
University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50208991(CHEMBL3884233)
Affinity DataIC50:  158nMAssay Description:Inhibition of biotin labelled VEGF165 binding to rat recombinant NRP-1/Fc chimeric protein incubated for overnight by competitive ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropilin-1(Rattus norvegicus)
University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50208991(CHEMBL3884233)
Affinity DataIC50:  160nMAssay Description:Inhibition of biotin labelled VEGF165 binding to rat recombinant NRP-1/Fc chimeric protein incubated for overnight by competitive ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropilin-1(Rattus norvegicus)
University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50167322(CHEMBL3799068)
Affinity DataIC50:  180nMAssay Description:Inhibition of (bt)-VEGF165 binding to purified recombinant rat NRP1/Fc chimera measured after overnight incubation by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Mossakowski Medical Research Centre Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50081523((S)-2-Amino-N-((R)-1-{[((S)-1-hydrazinocarbonyl-2-...)
Affinity DataIC50:  230nMAssay Description:Displacement of [3H]DELT2 from DOR in Sprague-Dawley rat brain homogenate measured after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropilin-1(Rattus norvegicus)
University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50208993(CHEMBL3885318)
Affinity DataIC50:  890nMAssay Description:Inhibition of biotin labelled VEGF165 binding to rat recombinant NRP-1/Fc chimeric protein incubated for overnight by competitive ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropilin-1(Rattus norvegicus)
University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50208993(CHEMBL3885318)
Affinity DataIC50:  890nMAssay Description:Inhibition of biotin labelled VEGF165 binding to rat recombinant NRP-1/Fc chimeric protein incubated for overnight by competitive ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropilin-1(Rattus norvegicus)
University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50317441(ATWLPPR | CHEMBL1095672)
Affinity DataIC50:  5.86E+3nMAssay Description:Inhibition of (bt)-VEGF165 binding to purified recombinant rat NRP1/Fc chimera measured after overnight incubation by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropilin-1(Rattus norvegicus)
University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50208994(CHEMBL3884096)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of biotin labelled VEGF165 binding to rat recombinant NRP-1/Fc chimeric protein incubated for overnight by competitive ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropilin-1(Rattus norvegicus)
University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50208995(CHEMBL3885243)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of biotin labelled VEGF165 binding to rat recombinant NRP-1/Fc chimeric protein incubated for overnight by competitive ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropilin-1(Rattus norvegicus)
University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50208992(CHEMBL3884504)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of biotin labelled VEGF165 binding to rat recombinant NRP-1/Fc chimeric protein incubated for overnight by competitive ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed