Found 225 with Last Name = 'liskamp' and Initial = 'rm' 
Affinity DataKi: 1.30nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
Affinity DataKi: 20nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
Affinity DataKi: 25nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
Affinity DataKi: 340nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
Affinity DataKi: 540nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
Affinity DataKi: 1.22E+3nMpH: 7.4Assay Description:The inhibition of plasma kallikrein and coagulation factor FXII was assessed by incubating the proteases with bicyclic peptide (twofold dilutions) an...More data for this Ligand-Target Pair
Affinity DataIC50: 1.32nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.45nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.45nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Displacement of [125I]NDP-MSH from human melanocortin receptor-4 expressed in 293 HEK cellsMore data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 8nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Displacement of [111In-DOTA0,Tyr3]octreotide from SSTR2 receptor in rat AR42J cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]NDP-MSH from human melanocortin receptor-4 expressed in 293 HEK cellsMore data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 16nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Displacement of 4-methylumbelliferyl from non-lysosomal GBA2 by fluorometryMore data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 20nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]NDP-MSH from human melanocortin receptor-4 expressed in 293 HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 30nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 44nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [111In]-(17)] as radioligand in pH 7.2 buffer, for 1 h at 37 deg...More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 45nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer upon incubation for 1 ...More data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Bristol-Myers Squibb Medical Imaging
Curated by ChEMBL
Affinity DataIC50: 54nMpH: 7.2Assay Description:Inhibitory concentration against human leukotriene B4 receptor using competing agent [3H]-LTB4 as radioligand in pH 7.2 buffer, for 1 h at 37 degree ...More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Displacement of [125I]NDP-MSH from human melanocortin receptor-4 expressed in 293 HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Displacement of 4-methylumbelliferyl from non-lysosomal GBA2 by fluorometryMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Displacement of [125I]NDP-MSH from human melanocortin receptor-4 expressed in 293 HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Binding affinity for Syk tandem SH2 domain in surface plasmon resonance assay (SPR)More data for this Ligand-Target Pair
Affinity DataIC50: 106nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 119nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Effective concentration against human melanocortin receptor-3 expressed in 293 HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 129nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Binding affinity for Syk tandem SH2 domain in surface plasmon resonance assay (SPR)More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 148nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]NDP-MSH from human melanocortin receptor-4 expressed in 293 HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]NDP-MSH from human melanocortin receptor-4 expressed in 293 HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Effective concentration against human melanocortin receptor-3 expressed in 293 HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Displacement of [125I]NDP-MSH from human melanocortin receptor-4 expressed in 293 HEK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 162nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 168nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 168nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 182nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 186nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
