Compile Data Set for Download or QSAR
maximum 50k data
Found 109 with Last Name = 'liu' and Initial = 'ch'
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307192(5-Chloro-6-hydroxy-N-(2-morpholinoethyl)nicotinami...)
Affinity DataIC50:  45nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307191(5,6-Dichloro-N-(2-morpholinoethyl)nicotinamide | C...)
Affinity DataIC50:  84nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307204(5,6-Dichloro-N-(3-morpholinopropyl)nicotinamide | ...)
Affinity DataIC50:  100nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307188(6-Chloro-N-(2-morpholinoethyl)nicotinamide | CHEMB...)
Affinity DataIC50:  180nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307208(2-Bromo-N-(2-morpholinoethyl)nicotinamide | CHEMBL...)
Affinity DataIC50:  320nMAssay Description:Inhibition of MAOB in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307201(6-Chloro-N-(3-morpholinopropyl)nicotinamide | CHEM...)
Affinity DataIC50:  380nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307189(6-Hydroxy-N-(2-morpholinoethyl)nicotinamide | CHEM...)
Affinity DataIC50:  430nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307210(4-Chloro-N-(2-morpholinoethyl)nicotinamide | CHEMB...)
Affinity DataIC50:  750nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482070(CHEMBL1089130)
Affinity DataIC50:  844nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482064(CHEMBL1090240)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50094999(CHEMBL3590018)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50094991(CHEMBL3590010)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50094998(CHEMBL3590017)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307207(2-Chloro-N-(2-morpholinoethyl)nicotinamide | CHEMB...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of MAOB in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482083(CHEMBL1089129)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307195(2-Bromo-N-(3-morpholinopropyl)nicotinamide | CHEMB...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of MAOB in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50095007(CHEMBL3590026)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50094990(CHEMBL3590009)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50095006(CHEMBL3590025)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307207(2-Chloro-N-(2-morpholinoethyl)nicotinamide | CHEMB...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  2.62E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50094996(CHEMBL3590015)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50094997(CHEMBL3590016)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50094982(CHEMBL3590007)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50094984(CHEMBL3590008)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482065(CHEMBL1091660)
Affinity DataIC50:  4.72E+3nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482081(CHEMBL1091179)
Affinity DataIC50:  4.72E+3nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM29136(CHEMBL92401 | Euphozid | Iprazid | Iproniazid)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50095004(CHEMBL3590023)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50095005(CHEMBL3590024)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307194(2-Chloro-N-(3-morpholinopropyl)nicotinamide | CHEM...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of MAOB in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482071(CHEMBL1091178)
Affinity DataIC50:  6.79E+3nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM15613(4-chloro-N-(2-morpholin-4-ylethyl)benzamide | 4-ch...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307197(4-Chloro-N-(3-morpholinopropyl)nicotinamide | CHEM...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM29136(CHEMBL92401 | Euphozid | Iprazid | Iproniazid)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of MAOB in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50094995(CHEMBL3590014)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307208(2-Bromo-N-(2-morpholinoethyl)nicotinamide | CHEMBL...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307194(2-Chloro-N-(3-morpholinopropyl)nicotinamide | CHEM...)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482087(CHEMBL1091941)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307205(5-Chloro-6-hydroxy-N-(3-morpholinopropyl)nicotinam...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482066(CHEMBL1091943)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50307187(6-Fluoro-N-(2-morpholinoethyl)nicotinamide | CHEMB...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of MAOA in Sprague-Dawley rat brain mitochondria using kynuramine substrate by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50094981(CHEMBL3590006)
Affinity DataIC50:  1.59E+4nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482069(CHEMBL1089128)
Affinity DataIC50:  1.59E+4nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482063(CHEMBL1090221)
Affinity DataIC50:  1.61E+4nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482068(CHEMBL1092197)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482079(CHEMBL1090219)
Affinity DataIC50:  1.72E+4nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1/Tubulin beta-2B chain(Bos taurus)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50095003(CHEMBL3590022)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of bovine brain tubulin polymerization extent after 20 mins by turbidimetricallyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50482085(CHEMBL1089884)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibition of Escherichia coli KAS3 after 1 min assessed as incorporation of 3H signal in the final product by liquid scintillation counterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 109 total ) | Next | Last >>
Jump to: