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Found 137 with Last Name = 'liu' and Initial = 'yq'
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518668(CHEMBL4546569)
Affinity DataIC50:  32nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518676(CHEMBL4453888)
Affinity DataIC50:  94nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067478(CHEMBL3400659)
Affinity DataIC50:  140nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518675(CHEMBL4458898)
Affinity DataIC50:  280nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518679(CHEMBL4468962)
Affinity DataIC50:  640nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518673(CHEMBL4448964)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518665(CHEMBL4445587)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518667(CHEMBL4585746)
Affinity DataIC50:  1.94E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518661(CHEMBL4554148)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518666(CHEMBL4556590)
Affinity DataIC50:  2.79E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518671(CHEMBL4560122)
Affinity DataIC50:  3.24E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518680(CHEMBL4573946)
Affinity DataIC50:  4.05E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518677(CHEMBL4467680)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518664(CHEMBL4473863)
Affinity DataIC50:  5.41E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518678(CHEMBL4516802)
Affinity DataIC50:  6.38E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM37953(US10093631, Compound Lesinurad | US10336710, Lesin...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM37953(US10093631, Compound Lesinurad | US10336710, Lesin...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of human URAT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067478(CHEMBL3400659)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518662(CHEMBL4436938)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518663(CHEMBL4551589)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518670(CHEMBL4568207)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518669(CHEMBL4517057)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067483(CHEMBL2375787)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067490(CHEMBL3400662)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067490(CHEMBL3400662)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067486(CHEMBL2375786)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067481(CHEMBL3400661)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067481(CHEMBL3400661)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067477(CHEMBL3400658)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067477(CHEMBL3400658)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067480(CHEMBL3400660)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067480(CHEMBL3400660)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant COX2 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067483(CHEMBL2375787)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50067486(CHEMBL2375786)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Hunan University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  7.84E+4nMAssay Description:Inhibition of ovine COX1 using fluorometric substrate after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518672(CHEMBL4594032)
Affinity DataIC50:  1.19E+5nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260319(CHEMBL4104534)
Affinity DataIC50:  2.34E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
Tianjin Medical University

Curated by ChEMBL
LigandPNGBDBM50518674(CHEMBL4459618)
Affinity DataIC50:  3.65E+5nMAssay Description:Inhibition of human URAT1 expressed in HEK293 cells assessed as reduction in [8-14C]uric acid uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260318(CHEMBL4061404)
Affinity DataIC50:  3.93E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260307(CHEMBL4089550)
Affinity DataIC50:  4.18E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260320(CHEMBL4094380)
Affinity DataIC50:  5.25E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260302(CHEMBL4064304)
Affinity DataIC50:  5.43E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260299(CHEMBL4088294)
Affinity DataIC50:  5.59E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260309(CHEMBL4077866)
Affinity DataIC50:  5.68E+5nMAssay Description:Reactivation of sarin-induced inhibition of human AChE assessed as dissociation constant using acetylthiocholine as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260313(CHEMBL4100639)
Affinity DataIC50:  6.26E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260308(CHEMBL4102122)
Affinity DataIC50:  6.37E+5nMAssay Description:Reactivation of VX-induced inhibition of human AChE assessed as dissociation constant using acetylthiocholine as substrate preincubated for 30 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260310(CHEMBL4064154)
Affinity DataIC50:  6.58E+5nMAssay Description:Reactivation of tabun-induced inhibition of human AChE assessed as dissociation constant using acetylthiocholine as substrate preincubated for 30 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50035852(HI-6)
Affinity DataIC50:  6.68E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Fourth Military Medical University

Curated by ChEMBL
LigandPNGBDBM50260322(CHEMBL4063109)
Affinity DataIC50:  6.85E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine as substrate preincubated for 30 mins followed by substrate addition measured every 5 mins for 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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