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Found 325 with Last Name = 'locatelli' and Initial = 'a'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187566(4-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzam...)
Affinity DataKi:  400nMAssay Description:Binding affinity to human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224371(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(e...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145415(1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(methylth...)
Affinity DataKi:  500nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142887(1-(tert-butyl)-3-(4-chlorophenyl)-4-aminopyrazolo[...)
Affinity DataKi:  500nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187569(4-(4-iodobenzylidene)-1-(4-iodophenyl)pyrazolidine...)
Affinity DataKi:  500nMAssay Description:Binding affinity to human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187573(3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-a...)
Affinity DataKi:  500nMAssay Description:Binding affinity to human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142887(1-(tert-butyl)-3-(4-chlorophenyl)-4-aminopyrazolo[...)
Affinity DataKi:  500nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187573(3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-a...)
Affinity DataKi:  500nMAssay Description:Binding affinity to human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187579(4-((6-bromobenzo[d][1,3]dioxol-5-yl)methylene)-1-(...)
Affinity DataKi:  500nMAssay Description:Binding affinity to human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142882(Butyl-[1-(2-chloro-2-phenyl-ethyl)-6-ethylsulfanyl...)
Affinity DataKi:  600nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187575(4-benzylidene-1-(4-iodophenyl)pyrazolidine-3,5-dio...)
Affinity DataKi:  600nMAssay Description:Binding affinity to human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224368(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(m...)
Affinity DataKi:  600nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142880(1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenet...)
Affinity DataKi:  700nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145425(1-(2-chloro-2-phenylethyl)-6-(ethylthio)-N-propyl-...)
Affinity DataKi:  700nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142880(1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenet...)
Affinity DataKi:  700nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187569(4-(4-iodobenzylidene)-1-(4-iodophenyl)pyrazolidine...)
Affinity DataKi:  800nMAssay Description:Binding affinity to human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50183364(1-(2-bromo-2-phenylethyl)-N-propyl-1H-pyrazolo[3,4...)
Affinity DataKi:  900nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187570(4-(2-(benzyloxy)benzylidene)-1-phenylpyrazolidine-...)
Affinity DataKi:  900nMAssay Description:Binding affinity to human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187574(4-((5-(3-chloro-4-methylphenyl)furan-2-yl)methylen...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187572(4-(3-(benzyloxy)benzylidene)-1-(3,4-dichlorophenyl...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187577(4-(4-(diethylamino)-2-hydroxybenzylidene)-1-(4-iod...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224376(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(p...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224385(1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenyl...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187568(2,4-dichloro-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)...)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity to human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187565(2-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzam...)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity to human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224381(1-(2-chloro-2-phenylethyl)-N-(3-fluorophenyl)-6-(m...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50183338(1-(2-bromo-2-phenylethyl)-4-(piperidin-1-yl)-1H-py...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142889(Butyl-[1-(2-chloro-2-phenyl-ethyl)-6-methylsulfany...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224388(CHEMBL238561 | N-(3-bromophenyl)-1-(2-chloro-2-phe...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187576(BAS-4844343 | CHEMBL207672 | N-(5-((1H-indol-3-yl)...)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity to human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187571(2-methoxy-4-(methylthio)-N-(5-phenethyl-1,3,4-thia...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187565(2-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzam...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50183347(2-(4-(phenethylamino)-1H-pyrazolo[3,4-d]pyrimidin-...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50183356(CHEMBL203492 | N-benzyl-1-styryl-1H-pyrazolo[3,4-d...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50183355(2-(4-(benzylamino)-1H-pyrazolo[3,4-d]pyrimidin-1-y...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142884(1-(2-Chloro-2-phenyl-ethyl)-6-methylsulfanyl-4-pip...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187579(4-((6-bromobenzo[d][1,3]dioxol-5-yl)methylene)-1-(...)
Affinity DataKi:  2.50E+3nMAssay Description:Binding affinity to human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50183345(1-(2-bromo-2-phenylethyl)-N-(2-ethoxyethyl)-1H-pyr...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50183351(1-(2-bromo-2-phenylethyl)-N-isopropyl-1H-pyrazolo[...)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224383(1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio...)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50183336(1-(2-bromo-2-phenylethyl)-N-butyl-1H-pyrazolo[3,4-...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50187578(BAS-0338868 | CHEMBL378903 | N-(5-phenethyl-1,3,4-...)
Affinity DataKi:  2.90E+3nMAssay Description:Binding affinity to human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50145411(1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-propyl...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224374(CHEMBL241749 | N-benzyl-1-(2-chloro-2-(4-chlorophe...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224387(1-(2-chloro-2-phenylethyl)-N-(2-chlorobenzyl)-6-(m...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50183342(CHEMBL382153 | N-benzyl-1-(2-bromo-2-phenylethyl)-...)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142890(1-(2-Chloro-2-phenyl-ethyl)-6-ethylsulfanyl-4-morp...)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142885(Benzyl-[1-(2-chloro-2-phenyl-ethyl)-6-methylsulfan...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibitory activity against Src in cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50142885(Benzyl-[1-(2-chloro-2-phenyl-ethyl)-6-methylsulfan...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50224366(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-1H-p...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of human recombinant SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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