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Found 149 with Last Name = 'lundström' and Initial = 'j'
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374091(CHEMBL257000)
Affinity DataIC50:  0.400nMAssay Description:Antagonist activity at CCR5 receptor by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323659(CHEMBL1208890 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  1nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323660(CHEMBL1208891 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  2nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377234(CHEMBL402902)
Affinity DataIC50:  3nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374084(CHEMBL257081)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374072(CHEMBL272716)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377234(CHEMBL402902)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of GSK3alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377237(CHEMBL255735)
Affinity DataIC50:  7nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377235(CHEMBL402541)
Affinity DataIC50:  9nMAssay Description:Inhibition of GSK3alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377235(CHEMBL402541)
Affinity DataIC50:  13nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377237(CHEMBL255735)
Affinity DataIC50:  13nMAssay Description:Inhibition of GSK3alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323662(CHEMBL1208954 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  13nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50274366(2-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-N-(4-(2-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374080(CHEMBL271075)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  17nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  17nMAssay Description:Inhibition of human p38-alpha kinase phosphorylationMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50274368(2-(5-tert-butyl-2-methylfuran-3-yl)-N-(4-(6-(morph...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human p38alpha phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377240(CHEMBL404565)
Affinity DataIC50:  20nMAssay Description:Inhibition of GSK3alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374087(CHEMBL272490)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323668(CHEMBL1208953 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  21nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50274367(2-(5-tert-butyl-2-methylfuran-3-yl)-N-(4-(2-morpho...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323666(CHEMBL1209013 | N-(5-tert-butyl-3-cyano-2-methoxyp...)
Affinity DataIC50:  22nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374798(CHEMBL255410)
Affinity DataIC50:  23nMAssay Description:Inhibition of human p38-alpha kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377232(CHEMBL253956)
Affinity DataIC50:  23nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377232(CHEMBL253956)
Affinity DataIC50:  23nMAssay Description:Inhibition of GSK3alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377240(CHEMBL404565)
Affinity DataIC50:  24nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323660(CHEMBL1208891 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  25nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377231(CHEMBL253748)
Affinity DataIC50:  26nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374082(CHEMBL402242)
Affinity DataIC50:  27nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323650(CHEMBL1209838 | N-(3-cyano-5-morpholinophenyl)-2-(...)
Affinity DataIC50:  28nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374074(CHEMBL257728)
Affinity DataIC50:  29nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM15244(5-(2,6-dichlorophenyl)-2-(2,4-difluorophenyl)sulfa...)
Affinity DataIC50:  29nMAssay Description:Inhibition of human p38-alpha kinaseMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374090(CHEMBL256584)
Affinity DataIC50:  31nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377241(CHEMBL402932)
Affinity DataIC50:  32nMAssay Description:Inhibition of GSK3alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323649(CHEMBL1209837 | N-(3-tert-butyl-5-cyanophenyl)-2-(...)
Affinity DataIC50:  33nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377231(CHEMBL253748)
Affinity DataIC50:  34nMAssay Description:Inhibition of GSK3alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323654(CHEMBL1208829 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  38nMAssay Description:Inhibition of phospho-p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377252(CHEMBL404175)
Affinity DataIC50:  38nMAssay Description:Inhibition of GSK3alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323662(CHEMBL1208954 | N-(5-tert-butyl-2-methoxy-3-(methy...)
Affinity DataIC50:  38nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  39nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  39nMAssay Description:Inhibition of human p38-alpha kinaseMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377248(CHEMBL255905)
Affinity DataIC50:  41nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323651(CHEMBL1209839 | N-(5-tert-butyl-3-cyano-2-methoxyp...)
Affinity DataIC50:  42nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  44nMAssay Description:Inhibition of human p38-alpha kinaseMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)
Affinity DataIC50:  44nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374078(CHEMBL272064)
Affinity DataIC50:  48nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377241(CHEMBL402932)
Affinity DataIC50:  49nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50323661(CHEMBL1208952 | N-(5-tert-butyl-3-cyano-2-methoxyp...)
Affinity DataIC50:  51nMAssay Description:Inhibition of p38 alpha activity by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kemia

Curated by ChEMBL
LigandPNGBDBM50377253(CHEMBL257575)
Affinity DataIC50:  51nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374073(CHEMBL255854)
Affinity DataIC50:  53nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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