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Found 1468 with Last Name = 'madan' and Initial = 'a'
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50005397(CHEMBL2206684)
Affinity DataKi:  0nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402366(CHEMBL2206696)
Affinity DataKi:  0.00100nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50005398(CHEMBL2206694)
Affinity DataKi:  0.00100nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402360(CHEMBL2206681)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402361(CHEMBL2206680)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402378(CHEMBL2206685)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402373(CHEMBL2206691)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402372(CHEMBL2206692)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402374(CHEMBL2206690)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402371(CHEMBL2206693)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402362(CHEMBL2206700)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402363(CHEMBL2206699)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402375(CHEMBL2206689)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402370(CHEMBL2206683)
Affinity DataKi:  0.00600nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402367(CHEMBL2206695)
Affinity DataKi:  0.00700nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402376(CHEMBL2206688)
Affinity DataKi:  0.00800nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402364(CHEMBL2206698)
Affinity DataKi:  0.0110nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402365(CHEMBL2206697)
Affinity DataKi:  0.0120nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402377(CHEMBL2206687)
Affinity DataKi:  0.0330nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50297306(CHEMBL540982 | {2-[3-(4-Fluoro-benzyl)-benzo[b]thi...)
Affinity DataKi:  0.0900nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in HEK293 Flp-In cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50297304(CHEMBL560741 | {2-[3-(4-Fluoro-benzyl)-1H-inden-2-...)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in HEK293 Flp-In cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402379(CHEMBL2206686)
Affinity DataKi:  0.296nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50315206((R)-2-(6-fluoro-3-(1-(thiazol-2-yl)ethyl)-1H-inden...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity at histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50297310((-)-Dimethyl-{2-[3-((R)-1-pyridin-2-yl-ethyl)-benz...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]N-methylscopolamine from human muscarinic M1 receptor expressed in CHO Flp-In cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50297307(CHEMBL564226 | R-dimethindene)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO Flp-In cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50316938(1-(4-fluorobenzyl)-2-(1-methylpiperidin-3-yl)-1H-b...)
Affinity DataKi:  0.5nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50261243((R)-1-(2-fluoro-6-(trifluoromethyl)benzyl)-3-(2-am...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I-Tyr5,DLeu6,NMeLeu7,Pro9-NEt-]GnRH from human GnRH receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50162007((R)-1-(2,6-difluorobenzyl)-3-(2-amino-2-phenylethy...)
Affinity DataKi:  0.560nMAssay Description:Displacement of [125I-Tyr5,DLeu6,NMeLeu7,Pro9-NEt-]GnRH from human GnRH receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50166450((R)-1-(2-fluoro-6-(trifluoromethyl)benzyl)-3-(2-am...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]Pro-N-Et-GnRH from human cloned GnRH receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50297305(CHEMBL559251 | Dimethyl-[2-(3-pyrazin-2ylmethyl-1H...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in HEK293 Flp-In cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188823(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50224184(1-{2-[(1S)-(3-dimethylaminopropionyl)amino-2-methy...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]NDP-MSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50221119(CHEMBL236521 | N-((S)-1-(2-(4-((R)-3-(2,4-dichloro...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]NDPMSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50297304(CHEMBL560741 | {2-[3-(4-Fluoro-benzyl)-1H-inden-2-...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]pyrilamine from human histamine H1 receptor expressed in CHO Flp-In cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50166450((R)-1-(2-fluoro-6-(trifluoromethyl)benzyl)-3-(2-am...)
Affinity DataKi:  0.640nMAssay Description:Displacement of [125I-Tyr5,DLeu6,NMeLeu7,Pro9-NEt-]GnRH from human GnRH receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50166450((R)-1-(2-fluoro-6-(trifluoromethyl)benzyl)-3-(2-am...)
Affinity DataKi:  0.640nMAssay Description:Binding affinity to human GnRHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50315205((R)-2-(6-fluoro-3-(1-(3-methoxypyrazin-2-yl)ethyl)...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190927(CHEMBL214513 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50315205((R)-2-(6-fluoro-3-(1-(3-methoxypyrazin-2-yl)ethyl)...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity at histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50221120(1-((R)-1-(4-(2-((S)-1-(2-aminoethylamino)-3-methyl...)
Affinity DataKi:  0.710nMAssay Description:Binding affinity to mouse MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50314264((-)-(R)-2-(1-(2-(2-(azetidin-1-yl)ethyl)benzo[b]th...)
Affinity DataKi:  0.730nMAssay Description:Inhibition of human ERG expressed in HEK cells assessed as blockade of potassium tail current by standard patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214688(1-{4-[(1R)-2-(amino-3-methylbutyl)-6-fluorophenyl]...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50214682(1-{4-[(1S)-2-(1-amino-3-methylbutyl)-4-trifluorome...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]NDP-MSH from MC4R receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50361005(CHEMBL1935442)
Affinity DataKi:  0.800nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50315198(2-(6-fluoro-3-((3-methoxypyrazin-2-yl)methyl)-1H-i...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity at histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50316936(2-(1-methylpiperidin-3-yl)-1-(2-phenoxyethyl)-1H-b...)
Affinity DataKi:  0.800nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50315191((R)-N,N-dimethyl-2-(3-(1-(thiazol-2-yl)ethyl)-1H-i...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity at histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50221120(1-((R)-1-(4-(2-((S)-1-(2-aminoethylamino)-3-methyl...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]NDPMSH from human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50166451((R)-1-(2-fluoro-6-(methylsulfonyl)benzyl)-3-(2-ami...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human GnRHRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190919(CHEMBL386454 | N-((S)-1-((R)-3-(4,4-dimethylcycloh...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to MCHR1 by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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