Affinity DataKi: 0.780nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17.6nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 273nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 706nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 863nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.43E+3nMAssay Description:Displacement of [3H]MRS2270 from human P2Y1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Antagonist activity against Turkey erythrocyte P2Y purinoceptor 1 (P2Y1) by the compound is measuredMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeSADP-induced inositol phosphate formationMore data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeS-ADP-stimulated PLC activityMore data for this Ligand-Target Pair
Affinity DataIC50: 157nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 206nMAssay Description:Antagonist activity against Turkey erythrocyte P2Y purinoceptor 1 (P2Y1) by the compound is measuredMore data for this Ligand-Target Pair
Affinity DataIC50: 221nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 356nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 367nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 377nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 452nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 617nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeS-ADP-stimulated PLC activityMore data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeSADP-induced inositol phosphate formationMore data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeSADP-induced inositol phosphate formationMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeS-ADP-stimulated PLC activityMore data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeSADP-induced inositol phosphate formationMore data for this Ligand-Target Pair
Affinity DataIC50: 871nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeS-ADP-stimulated PLC activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.55E+3nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeS-ADP-stimulated PLC activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+3nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeSADP-induced inositol phosphate formationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.74E+3nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeS-ADP-stimulated PLC activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.75E+3nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeSADP-induced inositol phosphate formationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.87E+3nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 1.94E+3nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeSADP-induced inositol phosphate formationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.95E+3nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeS-ADP-stimulated PLC activityMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair