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Found 388 with Last Name = 'manne' and Initial = 'v'
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405943(CHEMBL176596)
Affinity DataKi:  96nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405931(CHEMBL367753)
Affinity DataKi:  100nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405937(CHEMBL173782)
Affinity DataKi:  180nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405942(CHEMBL175345)
Affinity DataKi:  630nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405939(CHEMBL175307)
Affinity DataKi:  1.00E+3nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50018055(7-Amino-heptan-2-one | CHEMBL176843)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405932(CHEMBL176530)
Affinity DataKi:  2.60E+4nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405935(CHEMBL177305)
Affinity DataKi:  3.10E+4nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405928(CHEMBL174669)
Affinity DataKi:  7.50E+4nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405940(CHEMBL177890)
Affinity DataKi:  1.10E+5nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405930(CHEMBL174887)
Affinity DataKi:  1.30E+5nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405934(CHEMBL176764)
Affinity DataKi:  2.60E+5nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405929(CHEMBL436093)
Affinity DataKi:  3.76E+5nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405941(CHEMBL177777)
Affinity DataKi:  6.50E+5nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405938(CHEMBL81241)
Affinity DataKi:  8.00E+5nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405933(CHEMBL176800)
Affinity DataKi:  1.37E+6nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisomal N(1)-acetyl-spermine/spermidine oxidase(Homo sapiens (Human))
University Of The Pacific

Curated by ChEMBL
LigandPNGBDBM50405936(CHEMBL177217)
Affinity DataKi:  2.90E+7nMAssay Description:Ability to inhibit the deacetylation of [acetyl-3H]-N8-Acetylspermidine deacetylase in rat liver.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM13320(1-Methyl-1H-imidazole-4-sulfonic Acid [6-Cyano-1-(...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048982((R)-2-({(R)-2-[(R)-2-((S)-2-Amino-3-mercapto-propi...)
Affinity DataIC50:  0.370nMAssay Description:In vitro inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048970((R)-2-({(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propy...)
Affinity DataIC50:  0.460nMAssay Description:In vitro inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048963((R)-2-({(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propy...)
Affinity DataIC50:  0.570nMAssay Description:In vitro inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM13319(BMS-386914 | CHEMBL183536 | [[6-Cyano-1-(3-methyl-...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50164021(1-Methyl-1H-imidazole-4-sulfonic acid [6-cyano-1-(...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048972((R)-2-({(R)-2-[(R)-2-((S)-2-Amino-3-mercapto-propy...)
Affinity DataIC50:  0.600nMAssay Description:In vitro inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50085469((S)-2-({2-[(S)-2-((R)-2-Amino-3-mercapto-propylami...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50164025(BMS-316810 | CHEMBL360330 | Pyridine-2-sulfonic ac...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50164027(1-Methyl-1H-pyrazole-4-sulfonic acid [6-cyano-1-(3...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048967((R)-2-({(R)-2-[(R)-2-((S)-2-Amino-3-mercapto-propy...)
Affinity DataIC50:  0.75nMAssay Description:In vitro inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048399((S)-2-[((S)-2-{(S)-2-[2-(3H-Imidazol-4-yl)-ethylam...)
Affinity DataIC50:  0.790nMAssay Description:Inhibition of FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048399((S)-2-[((S)-2-{(S)-2-[2-(3H-Imidazol-4-yl)-ethylam...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50164003(CHEMBL183773 | N-[6-Cyano-1-(3-methyl-3H-imidazol-...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50164023(CHEMBL180307 | Pyridine-3-sulfonic acid [6-cyano-1...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50164017(CHEMBL183544 | N-[6-Cyano-1-(3-methyl-3H-imidazol-...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50164009(CHEMBL182813 | Pyridine-2-sulfonic acid [6-cyano-1...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50164013(CHEMBL439846 | Pyridine-3-sulfonic acid benzyl-[6-...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048964((R)-2-({(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propy...)
Affinity DataIC50:  0.920nMAssay Description:In vitro inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28030(2-aminopyridine analogue, 9 | N-{4-[(2-amino-3-chl...)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed using baculovirus expressed GST-Met, and poly(Glu/Tyr) as the substrate in the presence of test compound. Dose response c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048981((S)-2-({(R)-2-[(S)-2-((R)-3-Mercapto-2-methyl-prop...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28028(2-aminopyridine analogue, 7 | N-{4-[(2-amino-3-eth...)
Affinity DataIC50:  1nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed using baculovirus expressed GST-Met, and poly(Glu/Tyr) as the substrate in the presence of test compound. Dose response c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM13323(1-Methyl-1H-imidazole-4-sulfonic Acid Benzyl-[6-cy...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50370480(CHEMBL1169541)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50164012(CHEMBL183217 | Pyridine-3-sulfonic acid [6-cyano-1...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048966((R)-2-({(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propy...)
Affinity DataIC50:  1.30nMAssay Description:In vitro inhibition of Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM24457(2-[(3-fluoro-4-{1H-pyrrolo[2,3-b]pyridin-4-yloxy}p...)
Affinity DataIC50:  1.30nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed using baculovirus expressed GST-Met, and poly(Glu/Tyr) as the substrate. Dose response curves were generated to determine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092365((R)-1-((1H-imidazol-5-yl)methyl)-3-benzyl-4-(thiop...)
Affinity DataIC50:  1.35nMAssay Description:Inhibition of purified recombinant human farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50048968((R)-2-({(S)-2-[(S)-2-((R)-2-Amino-3-mercapto-propy...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibitory activity against FarnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM50235550(1-(4-(5-((4-aminocyclohexylidene)methyl)pyrrolo[1,...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human recombinant c-Met expressed in insect cell-baculovirus expression systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50164016(CHEMBL179598 | [[6-Cyano-1-(3-methyl-3H-imidazol-4...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092366(3-Benzyl-4-(2-dimethylamino-ethanesulfonyl)-1-(3H-...)
Affinity DataIC50:  1.53nMAssay Description:Inhibition of purified recombinant human farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Protein farnesyltransferase subunit beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092377(4-Benzenesulfonyl-3-benzyl-1-(3H-imidazol-4-ylmeth...)
Affinity DataIC50:  1.77nMAssay Description:Inhibition of purified recombinant human farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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