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Found 243 with Last Name = 'marson' and Initial = 'cm'
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196604(CHEMBL217083 | N-hydroxy-7-(naphthalen-2-yloxy)hep...)
Affinity DataIC50:  0.900nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196608(7-(4-((4-chlorobenzyl)(methyl)amino)phenoxy)-N-hyd...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196600(7-(1H-indol-5-yloxy)-N-hydroxyheptanamide | CHEMBL...)
Affinity DataIC50:  3.60nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataIC50:  5nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113971(CHEMBL3605506)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196598(7-(4-(3-(1H-indol-3-yl)prop-1-en-2-ylamino)phenyl1...)
Affinity DataIC50:  6.20nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113963(CHEMBL3605502)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50437812(CHEMBL2407723)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50437809(CHEMBL2407717)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196605(7-(4-(2-(1H-indol-3-yl)acetamido)phenyl1H-indol-3-...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196603(7-(4-(2-(1H-indol-3-yl)acetamido)-2-fluorophenyl1H...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50437821(CHEMBL2407736)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196594(7-(4-((1H-indol-5-yl)methylamino)phenyl1H-indol-5-...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196597(CHEMBL384714 | N-hydroxy-7-(4-(methyl(pyridin-4-yl...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113960(CHEMBL3605415)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50437816(CHEMBL2407719)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196609(7-(4-(3-(1H-indol-3-yl)propanamido)phenyl1H-indol-...)
Affinity DataIC50:  16nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196607(7-(4-(3-(1H-indol-3-yl)-N-(pyridin-4-ylmethyl)prop...)
Affinity DataIC50:  16nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113964(CHEMBL3605508)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113969(CHEMBL3605499)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196602(7-(4-(dimethylamino)phenoxy)-N-hydroxyheptanamide ...)
Affinity DataIC50:  19nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113954(CHEMBL3605507)
Affinity DataIC50:  21nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM24624(CHEMBL272980 | MGCD-0103 | MGCD0103 | N-(2-aminoph...)
Affinity DataIC50:  22nMAssay Description:Inhibition of His-tagged recombinant HDAC2 (1 to 488 residues) (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM24624(CHEMBL272980 | MGCD-0103 | MGCD0103 | N-(2-aminoph...)
Affinity DataIC50:  22nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196593(CHEMBL387042 | N-hydroxy-7-(4-((3-hydroxy-5-(hydro...)
Affinity DataIC50:  22nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196596(8-(4-(2-(1H-indol-3-yl)acetamido)phenyl1H-indol-3-...)
Affinity DataIC50:  22nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196601(CHEMBL217778 | N-hydroxy-7-(4-(4-methoxyphenylsulf...)
Affinity DataIC50:  22nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50437813(CHEMBL2407722)
Affinity DataIC50:  23nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196606(7-(4-(2-(1H-indol-3-yl)acetamido)-3-fluorophenyl1H...)
Affinity DataIC50:  24nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113967(CHEMBL3605497)
Affinity DataIC50:  24nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50437822(CHEMBL2407735)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113972(CHEMBL3605500)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50437827(CHEMBL2407730)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113962(CHEMBL3605495)
Affinity DataIC50:  33nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113968(CHEMBL3605498)
Affinity DataIC50:  34nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113966(CHEMBL3605496)
Affinity DataIC50:  34nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113953(CHEMBL3605503)
Affinity DataIC50:  35nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50437814(CHEMBL2407721)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113959(CHEMBL3605416)
Affinity DataIC50:  38nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113965(CHEMBL3605494)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50475567(6-Benzenesulfonylhexanoic Acid Hydroxamide | CHEMB...)
Affinity DataIC50:  40nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50437826(CHEMBL2407731)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113958(CHEMBL3605501)
Affinity DataIC50:  41nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM24624(CHEMBL272980 | MGCD-0103 | MGCD0103 | N-(2-aminoph...)
Affinity DataIC50:  45nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50223405(CHEMBL316183)
Affinity DataIC50:  49nMAssay Description:Inhibition of histone deacetylase (HDAC) activity in HeLa cell nuclear extractMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50196595(6-(4-(2-(1H-indol-3-yl)acetamido)phenyl1H-indol-3-...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of histone deacetylase activity using HeLa cell nuclear extract as enzyme sourceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50437815(CHEMBL2407720)
Affinity DataIC50:  52nMAssay Description:Inhibition of recombinant HDAC3-NCoR1 (unknown origin) using MAL as substrate incubated for 3 hrs prior to substrate addition measured after 60 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113970(CHEMBL3605504)
Affinity DataIC50:  55nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50113957(CHEMBL3605492)
Affinity DataIC50:  56nMAssay Description:Inhibition of recombinant HDAC3/NCOR2 (unknown origin) pre-incubated for 3 hrs before substrate addition by homogeneous fluorogenic HDAC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Rattus norvegicus)
University College London

Curated by ChEMBL
LigandPNGBDBM50475570(6-Benzenesulfinylhexanoic Acid Hydroxamide | CHEMB...)
Affinity DataIC50:  60nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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