Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]methylspiperone from human low affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cells by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Displacement of [3H]methylspiperone from human low affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11.7nMAssay Description:Displacement of [3H]methylspiperone from human low affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]Ro 41-1049 from MAO-A in rat cerebral cortex by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of [3H]methylspiperone from human low affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]methylspiperone from human low affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cells by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cells by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cells by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cells by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cells by competition binding assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Displacement of [3H]Ro 41-1049 from MAO-A in rat cerebral cortex by competition binding assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 92nMAssay Description:Displacement of [3H]Ro 41-1049 from MAO-A in rat cerebral cortex by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 109nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Displacement of [3H]methylspiperone from human low affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Displacement of [3H]methylspiperone from human low affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cells by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 127nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cells by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cells by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 157nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 187nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 194nMAssay Description:Displacement of [3H]methylspiperone from human low affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Displacement of [3H]methylspiperone from human low affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Competitive inhibition of human coagulation factor 11a using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 371nMAssay Description:Displacement of [3H]methylspiperone from human low affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 456nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 574nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Competitive inhibition of human coagulation factor 11a using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 803nMAssay Description:Displacement of [3H]7-OH-DPAT from human high affinity Dopamine D2S receptor by competition binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Neurosearch Sweden
Curated by ChEMBL
Neurosearch Sweden
Curated by ChEMBL
Affinity DataKi: 827nMAssay Description:Displacement of [3H]imipramine from human SERT expressed in CHO cells by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Competitive inhibition of human APC using S-2366 as substrateMore data for this Ligand-Target Pair