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Found 44 with Last Name = 'mccullough' and Initial = 'bs'
Target14 kDa phosphohistidine phosphatase(Homo sapiens)
University Of Utah College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50442875(NORSTICTIC ACID)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibition of PHPT1 (unknown origin) assessed as inhibition constant measured up to 100 uM incubated up to 30 mins using DiFMUP as fluorogenic substr...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataKi:  1.30E+5nMAssay Description:Non-covalent inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 15 to 120 mins followed by substrate addition at pH 6.5 by st...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataKi:  1.30E+5nMAssay Description:Non-covalent inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 15 to 120 mins followed by substrate addition at pH 6.5 by st...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMediator of RNA polymerase II transcription subunit 25(Homo sapiens)
University Of Utah College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50442875(NORSTICTIC ACID)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of Med25 transcriptional activation in human MCF-7 cells by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target14 kDa phosphohistidine phosphatase(Homo sapiens)
University Of Utah College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50442875(NORSTICTIC ACID)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of PHPT1 (unknown origin) using DiFMUP as fluorogenic substrate incubated for 30 mins followed by substrate addition and measured every 60...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CD45 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CD45 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase mu(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of PTPmu (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase mu(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of PTPmu (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target14 kDa phosphohistidine phosphatase(Homo sapiens)
University Of Utah College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50056922(1,4-Dihydroxy-10-methoxy-5,8-dimethyl-3,7-dioxo-1,...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of PHPT1 (unknown origin) using DiFMUP as fluorogenic substrate incubated for 30 mins followed by substrate addition and measured every 60...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of SHP2 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of SHP2 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target14 kDa phosphohistidine phosphatase(Homo sapiens)
University Of Utah College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50239376(CHEBI:35817 | ROXARSONE)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of PHPT1 (unknown origin) using DiFMUP as fluorogenic substrate incubated for 30 mins followed by substrate addition and measured every 60...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of LMWPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TCPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase epsilon(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPep (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of LMWPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CD45 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HePTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase epsilon(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPep (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase epsilon(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPep (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target14 kDa phosphohistidine phosphatase(Homo sapiens)
University Of Utah College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50240028(Acetarsol | Acetarsone | Gynoplix | S.V.C. | Stova...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of PHPT1 (unknown origin) using DiFMUP as fluorogenic substrate incubated for 30 mins followed by substrate addition and measured every 60...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of VHR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HePTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TCPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of VHR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HePTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of SHP2 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase mu(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPmu (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CD45 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of LMWPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of VHR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TCPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of VHR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TCPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of SHP2 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase mu(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPmu (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50262987(CHEMBL506661 | Illudalic acid)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HePTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of LMWPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase epsilon(Homo sapiens (Human))
University of Utah

Curated by ChEMBL
LigandPNGBDBM50263036(3-Hydroxy-6-methoxy-8,8-dimethyl-1-oxo-1,3,4,7,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPep (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed