TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Inhibition of human DAGLalpha expressed in HEK293T cell membranes assessed as reduction in hydrolysis of inhibition of [14C]-sn-1-oleoyl-2-arachidono...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 794nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Inhibition of human ABHD6 expressed in HEK293T cell membranes assessed as reduction in glycerol production using 2-arachidonoyl glycerol substrateMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.26E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.59E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 1.59E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Inhibition of human ABHD6 expressed in HEK293T cell membranes assessed as reduction in glycerol production using 2-arachidonoyl glycerol substrateMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 6.31E+3nMAssay Description:Displacement of [3H]ZM241385 from human AA2AR expressed in HEK293T cells after 2 hrs by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 1.83E+4nMAssay Description:Inhibition of human ABHD6 expressed in HEK293T cell membranes assessed as reduction in glycerol production using 2-arachidonoyl glycerol substrateMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 2.51E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 3.98E+4nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Radboud University Nijmegen Medical Centre
Curated by ChEMBL
Affinity DataKi: 7.94E+5nMAssay Description:Displacement of [3H]dihydroalprenolol from human ADRB2 expressed in HEK293T cells after 1 hr by liquid scintillation counterMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human Glycine Transporter type-2More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human DAGLalpha expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of human DAGLalpha expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibition of human DAGLalpha expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Inhibition of human DAGLalpha expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Inhibition of human Glycine Transporter type-2More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibition of human Glycine Transporter type-2More data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:Inhibition of human DAGLalpha expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:In vitro inhibition of human Glycine Transporter type-1.More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:In vitro inhibition of human Glycine Transporter type-1.More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:In vitro inhibition of human Glycine Transporter type-1.More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:In vitro inhibition of human Glycine Transporter type-1.More data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Inhibition of MB064 labeling of DAGLalpha in mouse brain homogenates by activity based protein profiling assayMore data for this Ligand-Target Pair
Affinity DataIC50: 143nMAssay Description:Inhibition of human DAGLalpha expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 185nMAssay Description:Inhibition of human DAGLalpha expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Organon Research And Development Group
Curated by ChEMBL
Organon Research And Development Group
Curated by ChEMBL
Affinity DataIC50: 209nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
Organon Laboratories
Curated by ChEMBL
Organon Laboratories
Curated by ChEMBL
Affinity DataIC50: 214nMAssay Description:Inhibition of human Glycine Transporter type-2More data for this Ligand-Target Pair
Affinity DataIC50: 302nMAssay Description:Inhibition of human DAGLalpha expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Organon Research And Development Group
Curated by ChEMBL
Organon Research And Development Group
Curated by ChEMBL
Affinity DataIC50: 331nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Organon Research And Development Group
Curated by ChEMBL
Organon Research And Development Group
Curated by ChEMBL
Affinity DataIC50: 339nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Organon Research And Development Group
Curated by ChEMBL
Organon Research And Development Group
Curated by ChEMBL
Affinity DataIC50: 347nMAssay Description:Inhibition of HIV-1 reverse transcriptase (HIV-1 RT)More data for this Ligand-Target Pair
Affinity DataIC50: 355nMAssay Description:Inhibition of MB064 labeling of DAGLalpha in mouse brain homogenates by activity based protein profiling assayMore data for this Ligand-Target Pair