Affinity DataKi: 2.80nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor overexpressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor over-expressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor overexpressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor overexpressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
Affinity DataKd: 1.30nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 9.10nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 21nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 51nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 44nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 8.70nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 8.5nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 8.5nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 33nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 650nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 280nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 440nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 420nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 7.90nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 30nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 310nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 480nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 53nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 240nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 82nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 260nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 46nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 40nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 42nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 450nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
Affinity DataKd: 170nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
Affinity DataKd: 9.40nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
Affinity DataKd: 9.40nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 8.20E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential preincubat...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 390nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential preincubat...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 920nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential preincubat...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 8.48E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 1.25E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataEC50: 78nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair