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Found 100 with Last Name = 'melin' and Initial = 'p'
TargetOxytocin receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50403716(CHEMBL2112378)
Affinity DataKi:  2.80nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor overexpressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50081738(2-[(3S,6S,9S,12S,15R)-3-(3-Amino-propyl)-9-((R)-se...)
Affinity DataKi:  26nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor over-expressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50081738(2-[(3S,6S,9S,12S,15R)-3-(3-Amino-propyl)-9-((R)-se...)
Affinity DataKi:  26nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor overexpressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50403717(CHEMBL2112376)
Affinity DataKi:  1.00E+3nMAssay Description:In vivo antagonistic activity against cloned human oxytocin receptor overexpressed in a stable HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016310(CHEMBL406303 | [Mpa1Val4Sar7]AVP (Arginine-vasopre...)
Affinity DataKd:  1.30nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016312(CHEMBL265119 | [Sar7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  9.10nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016314(CHEMBL269715 | [MeAla7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  21nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016316(CHEMBL413706 | [Phe2MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  100nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016318(CHEMBL411357 | [Mpa1,MeAla7,D-Arg8]VP (Vasopressin...)
Affinity DataKd:  51nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016309(CHEMBL410025 | [Phe2Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  44nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016311(CHEMBL413249 | [Mpa1Sar7,Drg8]VP (Vasopressin ))
Affinity DataKd:  8.70nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016313(CHEMBL217517 | [Val4Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  8.5nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016317(CHEMBL2371674 | [Mpa1Val4MeAla7]AVP (Arginine-vaso...)
Affinity DataKd:  8.5nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016315(CHEMBL437631 | [Val4MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  33nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016312(CHEMBL265119 | [Sar7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  650nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016314(CHEMBL269715 | [MeAla7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  280nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016314(CHEMBL269715 | [MeAla7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  440nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016312(CHEMBL265119 | [Sar7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  10nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016312(CHEMBL265119 | [Sar7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  420nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016314(CHEMBL269715 | [MeAla7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  19nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016311(CHEMBL413249 | [Mpa1Sar7,Drg8]VP (Vasopressin ))
Affinity DataKd:  160nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016311(CHEMBL413249 | [Mpa1Sar7,Drg8]VP (Vasopressin ))
Affinity DataKd:  7.90nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016315(CHEMBL437631 | [Val4MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  30nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016315(CHEMBL437631 | [Val4MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  310nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016315(CHEMBL437631 | [Val4MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  480nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016317(CHEMBL2371674 | [Mpa1Val4MeAla7]AVP (Arginine-vaso...)
Affinity DataKd:  53nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016311(CHEMBL413249 | [Mpa1Sar7,Drg8]VP (Vasopressin ))
Affinity DataKd:  240nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016317(CHEMBL2371674 | [Mpa1Val4MeAla7]AVP (Arginine-vaso...)
Affinity DataKd:  82nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016309(CHEMBL410025 | [Phe2Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  170nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016318(CHEMBL411357 | [Mpa1,MeAla7,D-Arg8]VP (Vasopressin...)
Affinity DataKd:  290nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016309(CHEMBL410025 | [Phe2Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  260nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016318(CHEMBL411357 | [Mpa1,MeAla7,D-Arg8]VP (Vasopressin...)
Affinity DataKd:  46nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016309(CHEMBL410025 | [Phe2Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  40nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016310(CHEMBL406303 | [Mpa1Val4Sar7]AVP (Arginine-vasopre...)
Affinity DataKd:  42nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016316(CHEMBL413706 | [Phe2MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  110nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016316(CHEMBL413706 | [Phe2MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  170nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016310(CHEMBL406303 | [Mpa1Val4Sar7]AVP (Arginine-vasopre...)
Affinity DataKd:  27nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016310(CHEMBL406303 | [Mpa1Val4Sar7]AVP (Arginine-vasopre...)
Affinity DataKd:  1.40nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016316(CHEMBL413706 | [Phe2MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  110nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016318(CHEMBL411357 | [Mpa1,MeAla7,D-Arg8]VP (Vasopressin...)
Affinity DataKd:  450nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016313(CHEMBL217517 | [Val4Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  110nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016313(CHEMBL217517 | [Val4Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  170nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016313(CHEMBL217517 | [Val4Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  9.40nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016317(CHEMBL2371674 | [Mpa1Val4MeAla7]AVP (Arginine-vaso...)
Affinity DataKd:  9.40nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataEC50:  8.20E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential preincubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581833(CHEMBL1949980)
Affinity DataEC50:  390nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential preincubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581834(CHEMBL5080252)
Affinity DataEC50:  920nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataEC50:  8.48E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581833(CHEMBL1949980)
Affinity DataEC50:  1.25E+3nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50581834(CHEMBL5080252)
Affinity DataEC50:  78nMAssay Description:Potentiation of CFTR F508del mutant (unknown origin) expressed in CHO cells assessed as chloride transport by measuring membrane potential incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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