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Found 91 with Last Name = 'michelotti' and Initial = 'el'
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482992(CHEMBL1269927)
Affinity DataIC50:  8nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482992(CHEMBL1269927)
Affinity DataIC50:  47nMAssay Description:Inhibition of HIV1 reverse transcriptase L100I mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482991(CHEMBL1270036)
Affinity DataIC50:  55nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482991(CHEMBL1270036)
Affinity DataIC50:  70nMAssay Description:Inhibition of HIV1 reverse transcriptase L100I mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482996(CHEMBL1269928)
Affinity DataIC50:  70nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483013(CHEMBL1271250)
Affinity DataIC50:  70nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483007(CHEMBL1270035)
Affinity DataIC50:  80nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483008(CHEMBL1271460)
Affinity DataIC50:  83nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482995(CHEMBL1270141)
Affinity DataIC50:  90nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483009(CHEMBL1271251)
Affinity DataIC50:  90nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  290nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174086(CHEMBL198470 | N-(3-hydroxy-4-(1-hydroxy-2-methylp...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174085(CHEMBL198563 | N-(3-(trifluoromethyl)benzyl)-4-phe...)
Affinity DataIC50:  450nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483001(CHEMBL1271043)
Affinity DataIC50:  500nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174095(CHEMBL198832 | N-(3-(trifluoromethoxy)benzyl)-4-ph...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174098(CHEMBL197228 | N-((2,3-dihydro-1H-inden-5-yl)methy...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174090(CHEMBL199074 | N-(4-(trifluoromethyl)benzyl)-4-phe...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174097(4-phenoxy-N-(pyridin-2-ylmethyl)benzamide | CHEMBL...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174096(CHEMBL199174 | N-(4-methyl-benzyl)-4-phenoxy-benza...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174092(CHEMBL199229 | N-(3-hydroxy-4-(1-hydroxy-2-methylp...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482993(CHEMBL1270346)
Affinity DataIC50:  2.57E+3nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483003(CHEMBL1270839)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482998(CHEMBL1271352)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483006(CHEMBL1271148)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482999(CHEMBL1271351)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174088(4-(2-hydroxybenzylamino)-N-(3-(4-fluorophenoxy)phe...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482992(CHEMBL1269927)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482992(CHEMBL1269927)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482991(CHEMBL1270036)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase Y188L mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482994(CHEMBL1270142)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174100(4-(2-hydroxybenzylamino)-N-(3-(2,4-difluorophenoxy...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174089(4-(2-hydroxybenzylamino)-N-(3-phenoxyphenyl)piperi...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174094(4-(2-hydroxybenzylamino)-N-(3-(2-chlorophenoxy)phe...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174093(4-(2-hydroxybenzylamino)-N-(3-(3-(trifluoromethyl)...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174099(2-((1-(3-phenoxybenzylsulfonyl)piperidin-4-ylamino...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174087(4-(naphthalen-1-ylmethylamino)-N-(3-phenoxyphenyl)...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174091(4-(benzylamino)-N-(3-phenoxyphenyl)piperidine-1-su...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483005(CHEMBL1270245)
Affinity DataIC50:  2.36E+4nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482991(CHEMBL1270036)
Affinity DataIC50:  3.67E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483011(CHEMBL1270940)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483002(CHEMBL1270941)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483000(CHEMBL1271147)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50482997(CHEMBL1271459)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483004(CHEMBL1270345)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483012(CHEMBL1270246)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Ansaris

Curated by ChEMBL
LigandPNGBDBM50483010(CHEMBL1271044)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of wild type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin polymerization-promoting protein(Bos taurus)
Rohm And Haas

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataEC50:  750nMAssay Description:Inhibition of Bos taurus (bovine) brain tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin polymerization-promoting protein(Bos taurus)
Rohm And Haas

Curated by ChEMBL
LigandPNGBDBM50099938(((1S,6R)-6-Nitro-cyclohex-3-enyl)-benzene | CHEMBL...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of Bos taurus (bovine) brain tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin polymerization-promoting protein(Bos taurus)
Rohm And Haas

Curated by ChEMBL
LigandPNGBDBM50099944(1-Methoxy-3-((1S,6R)-6-nitro-cyclohex-3-enyl)-benz...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of Bos taurus (bovine) brain tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin polymerization-promoting protein(Bos taurus)
Rohm And Haas

Curated by ChEMBL
LigandPNGBDBM50099946(1,2,3-Trimethoxy-4-(6-nitro-cyclohex-3-enyl)-benze...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of Bos taurus (bovine) brain tubulin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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