Compile Data Set for Download or QSAR
maximum 50k data
Found 158 with Last Name = 'mikhail' and Initial = 'a'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50185040(CHEMBL204828 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197135(CHEMBL217442 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207679(CHEMBL246258 | N-(1-(2-chloro-4-((2-(pyrrolidin-1-...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197136(CHEMBL387178 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197143(CHEMBL277531 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197116(CHEMBL217706 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  2.5nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207681(CHEMBL248297 | N-(1-(3-fluoro-4-(3-(piperidin-1-yl...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197139(CHEMBL214021 | N-(1-(benzo[d][1,3]dioxol-5-ylmethy...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50185040(CHEMBL204828 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197144(CHEMBL387418 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197139(CHEMBL214021 | N-(1-(benzo[d][1,3]dioxol-5-ylmethy...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197111(CHEMBL213715 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  3.60nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197124(CHEMBL217789 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  3.60nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197113(CHEMBL214731 | N-(1-(benzo[d][1,3]dioxol-5-ylmethy...)
Affinity DataIC50:  4nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207674(CHEMBL245844 | N-(1-(4-(3-(2,4-dioxothiazolidin-3-...)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197124(CHEMBL217789 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197109(CHEMBL387417 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  5nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197120(CHEMBL217593 | N-[1-[(4-methoxybenzyl)methyl]piper...)
Affinity DataIC50:  5.40nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197137(CHEMBL217707 | N-[1-[(2,2-difluoro-1,3-benzodioxol...)
Affinity DataIC50:  5.60nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197136(CHEMBL387178 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  6.20nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197114(CHEMBL214767 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  6.70nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197131(CHEMBL214377 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  7.40nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197123(CHEMBL214768 | N-(1-(3-fluoro-4-methoxybenzyl)pipe...)
Affinity DataIC50:  8.5nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197108(CHEMBL217400 | N-[1-[(3-methoxybenzyl)methyl]piper...)
Affinity DataIC50:  10.4nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197144(CHEMBL387418 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  10.5nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50185042(CHEMBL206081 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  11nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50185042(CHEMBL206081 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  11.5nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197119(CHEMBL216225 | N-[1-[(3-fluorobenzyl)methyl]piperi...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197115(CHEMBL425448 | N-[1-[(2,3-dihydro-1,4-benzodioxin-...)
Affinity DataIC50:  12.2nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197120(CHEMBL217593 | N-[1-[(4-methoxybenzyl)methyl]piper...)
Affinity DataIC50:  13nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197136(CHEMBL387178 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at MCHr1 assessed as inhibition of MCH-mediated calcium ion release in intact IMR32 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197146(CHEMBL217105 | N-{1-[(6-chloro-1,3-benzodioxol-5-y...)
Affinity DataIC50:  13.5nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197129(CHEMBL387309 | N-[1-[(2-fluoro-4-methoxybenzyl)met...)
Affinity DataIC50:  14.7nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207685(CHEMBL394639 | N-(1-(3-fluoro-4-(2-(isobutoxyimino...)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197139(CHEMBL214021 | N-(1-(benzo[d][1,3]dioxol-5-ylmethy...)
Affinity DataIC50:  15.1nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197135(CHEMBL217442 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  15.9nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197135(CHEMBL217442 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at MCHr1 assessed as inhibition of MCH-mediated calcium ion release in intact IMR32 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207684(CHEMBL246050 | N-(1-(4-((2-(piperidin-1-yl)ethyl)c...)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197118(CHEMBL213761 | N-[1-benzylpiperidin-4-yl]-7-fluoro...)
Affinity DataIC50:  19.9nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207677(CHEMBL248296 | N-(1-(4-(3-(dimethylamino)propoxy)-...)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197132(CHEMBL384487 | N-[1-{4-[(4-aminopiperidin-1-yl)met...)
Affinity DataIC50:  20.3nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197119(CHEMBL216225 | N-[1-[(3-fluorobenzyl)methyl]piperi...)
Affinity DataIC50:  21.2nMAssay Description:Displacement of [3H]dofetilide from hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197146(CHEMBL217105 | N-{1-[(6-chloro-1,3-benzodioxol-5-y...)
Affinity DataIC50:  22nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207675(CHEMBL246464 | N-(1-(3-fluoro-4-(3-(piperidin-1-yl...)
Affinity DataIC50:  23nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197125(CHEMBL386021 | N-[1-(1,3-benzodioxol-5-ylmethyl)pi...)
Affinity DataIC50:  24nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197123(CHEMBL214768 | N-(1-(3-fluoro-4-methoxybenzyl)pipe...)
Affinity DataIC50:  24nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197123(CHEMBL214768 | N-(1-(3-fluoro-4-methoxybenzyl)pipe...)
Affinity DataIC50:  24nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207673(CHEMBL246259 | N-(1-(2-methoxy-4-((2-(pyrrolidin-1...)
Affinity DataIC50:  26nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207683(CHEMBL245846 | N-(1-(3-fluoro-4-((2-(pyrrolidin-1-...)
Affinity DataIC50:  29nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197139(CHEMBL214021 | N-(1-(benzo[d][1,3]dioxol-5-ylmethy...)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at MCHR1 assessed as inhibition of MCH-mediated calcium release in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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