Compile Data Set for Download or QSAR
maximum 50k data
Found 65 with Last Name = 'miller' and Initial = 'sg'
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374091(CHEMBL257000)
Affinity DataIC50:  0.400nMAssay Description:Antagonist activity at CCR5 receptor by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374072(CHEMBL272716)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374084(CHEMBL257081)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374080(CHEMBL271075)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374087(CHEMBL272490)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374082(CHEMBL402242)
Affinity DataIC50:  27nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374074(CHEMBL257728)
Affinity DataIC50:  29nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374090(CHEMBL256584)
Affinity DataIC50:  31nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374078(CHEMBL272064)
Affinity DataIC50:  48nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374073(CHEMBL255854)
Affinity DataIC50:  53nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374089(CHEMBL272556)
Affinity DataIC50:  78nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374075(CHEMBL402776)
Affinity DataIC50:  96nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374081(CHEMBL271076)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374088(CHEMBL411640)
Affinity DataIC50:  271nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374085(CHEMBL405634)
Affinity DataIC50:  271nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374076(CHEMBL256792)
Affinity DataIC50:  310nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374086(CHEMBL272581)
Affinity DataIC50:  323nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374083(CHEMBL255855)
Affinity DataIC50:  381nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374079(CHEMBL404056)
Affinity DataIC50:  539nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
K£Mia

Curated by ChEMBL
LigandPNGBDBM50374077(CHEMBL255535)
Affinity DataIC50:  970nMAssay Description:Displacement of [125I]MIP1beta from human recombinant CCR5 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105938(4-{N'-[1-(3,4-Dimethyl-phenyl)-3-ethoxy-5-oxo-1,5-...)
Affinity DataEC50:  600nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105936(3-Hydroxy-4-[N'-(3-methyl-5-oxo-1-phenyl-1,5-dihyd...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105937(3-Hydroxy-4-(10-hydroxy-phenanthren-9-ylazo)-napht...)
Affinity DataEC50:  200nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105939(3-Hydroxy-4-[N'-(3-methyl-5-oxo-1-o-tolyl-1,5-dihy...)
Affinity DataEC50:  1.00E+4nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105940(4-{N'-[1-(3,4-Dimethyl-phenyl)-5-oxo-1,5-dihydro-p...)
Affinity DataEC50:  100nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105942(4-{N'-[1-(3-tert-Butyl-phenyl)-3-methyl-5-oxo-1,5-...)
Affinity DataEC50:  70nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105944(3-Hydroxy-4-(2-hydroxy-5-methyl-phenylazo)-naphtha...)
Affinity DataEC50:  3.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105941(4-(2,3-Dihydroxy-naphthalen-1-ylazo)-3-hydroxy-nap...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105943(4-[N'-(1-Benzyl-3-methyl-5-oxo-1,5-dihydro-pyrazol...)
Affinity DataEC50: >3.00E+4nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105947(3-Hydroxy-4-{N'-[3-methyl-5-oxo-1-(3-trifluorometh...)
Affinity DataEC50:  40nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105946(4-{N'-[1-(3,4-Dimethyl-phenyl)-5-oxo-3-phenyl-1,5-...)
Affinity DataEC50:  900nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105948(4-{N'-[1-(3-Chloro-phenyl)-3-methyl-5-oxo-1,5-dihy...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105949(4-(2,4-Dihydroxy-naphthalen-1-ylazo)-3-hydroxy-nap...)
Affinity DataEC50:  5.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105951(4-(2,6-Dihydroxy-naphthalen-1-ylazo)-3-hydroxy-nap...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105952(4-{N'-[1-(4-Fluoro-phenyl)-3-methyl-5-oxo-1,5-dihy...)
Affinity DataEC50:  500nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105945(3-Hydroxy-4-[N'-(3-methyl-5-oxo-1-p-tolyl-1,5-dihy...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105956(3-Hydroxy-4-(2-hydroxy-4-sulfo-naphthalen-1-ylazo)...)
Affinity DataEC50:  1.00E+4nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105953(4-(2,7-Dihydroxy-naphthalen-1-ylazo)-3-hydroxy-nap...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105955(3-Hydroxy-4-{N'-[3-methyl-1-(2-nitro-phenyl)-5-oxo...)
Affinity DataEC50:  8.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105954(1-(4-tert-Butyl-phenyl)-4-[(2-hydroxy-4-sulfo-naph...)
Affinity DataEC50:  200nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105959(3-Hydroxy-4-{N'-[3-methyl-1-(4-nitro-phenyl)-5-oxo...)
Affinity DataEC50:  400nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105958(3-Hydroxy-4-[N'-(3-methyl-5-oxo-1-p-tolyl-1,5-dihy...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105950(4-{N'-[1-(3,4-Dichloro-phenyl)-3-methyl-5-oxo-1,5-...)
Affinity DataEC50:  200nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105957(4-{N'-[3-Amino-1-(4-tert-butyl-phenyl)-5-oxo-1,5-d...)
Affinity DataEC50:  5.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105962(3-Hydroxy-4-{N'-[1-(4-isopropyl-phenyl)-3-methyl-5...)
Affinity DataEC50:  70nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105960(3-Hydroxy-4-[N'-(3-methyl-5-oxo-1-m-tolyl-1,5-dihy...)
Affinity DataEC50:  700nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105961(3-Hydroxy-4-(2-hydroxy-7-methoxy-naphthalen-1-ylaz...)
Affinity DataEC50:  300nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105964(3-Hydroxy-4-[N'-(3-methyl-5-oxo-1-pyridin-2-yl-1,5...)
Affinity DataEC50:  7.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105967(3-Hydroxy-4-{N'-[1-(4-iodo-phenyl)-3-methyl-5-oxo-...)
Affinity DataEC50:  300nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThrombopoietin receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50105965(4-{N'-[1-(3,4-Dimethyl-phenyl)-3-methyl-5-oxo-1,5-...)
Affinity DataEC50:  1.00E+3nMAssay Description:Effective concentration for thrombopoietin luciferase activity was determined in BAF-3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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