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Found 506 with Last Name = 'mort' and Initial = 'n'
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84707(nafarelin)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84726(deslorelin)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469862(CHEMBL409219)
Affinity DataKi:  0.0135nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84708(deslorelin 31Nal)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84712(deslorelin 2NMePhe | deslorelin 2Phe)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469858(CHEMBL268397)
Affinity DataKi:  0.0234nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84728(nafarelin 5NMeTyr)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84711(nafarelin 31Nal)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84717(nafarelin 7NMeLeu)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84703(nafarelin 10SarNH2)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469859(A-75998 | CHEMBL263839)
Affinity DataKi:  0.0316nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469856(CHEMBL263840 | ORG-30850)
Affinity DataKi:  0.0331nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84713(nafarelin 4NMeSer)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469857(CHEMBL268319)
Affinity DataKi:  0.0525nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84715(deslorelin 7NMeLeu)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469860(CHEMBL409990)
Affinity DataKi:  0.0617nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84730(nafarelin 2Phe)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84704(deslorelin 4NMeSer)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84700(leuprolide 31Nal)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84721(deslorelin 5NMeTyr)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50469861(CHEMBL438829)
Affinity DataKi:  0.117nMAssay Description:The negative logarithm of the concentration of antagonist that inhibits 50% of the binding of 125 I-labeled leuprolide to the rat pituitary LHRH rece...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84727(leuprolide 7NMeLeu)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84712(deslorelin 2NMePhe | deslorelin 2Phe)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84731(nafarelin 2NMePhe)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84714(deslorelin 8NMeArg)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84720(deslorelin 10SarNH2)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84702(nafarelin 3NMe1Nal)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84719(deslorelin 3NMe1Nal)
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84701(CAS_35263-73-1 | LHRH)
Affinity DataKi:  1.26nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84718(nafarelin 2NMeHis)
Affinity DataKi:  1.41nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84732(deslorelin 2NMeHis)
Affinity DataKi:  1.41nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84722(leuprolide 4NMeSer)
Affinity DataKi:  1.41nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84710(leuprolide 2 Phe)
Affinity DataKi:  2.19nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84724(leuprolide 5NMeTyr)
Affinity DataKi:  2.51nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84705(nafarelin 6NMe2Nal)
Affinity DataKi:  2.69nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84723(leuprolide 3NMe1Nal)
Affinity DataKi:  3.24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84729(leuprolide 6NMeDLeu)
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84706(leuprolide 10SarNH2)
Affinity DataKi:  10.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84733(leuprolide 2NMePhe)
Affinity DataKi:  12.0nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84709(nafarelin 8NMeArg)
Affinity DataKi:  28.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84699(leuprolide 2 NMeHis)
Affinity DataKi:  33.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgonadoliberin-1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM84716(leuprolide 8NMeArg)
Affinity DataKi:  347nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrans-sialidase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM50118216((4-formyl-5-hydroxy-6-methylpyridin-3-yl)methyl di...)
Affinity DataKi:  7.30E+6nMAssay Description:Inhibition of Trypanosoma cruzi trans-SialidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrans-sialidase(Trypanosoma cruzi)
University Of Manchester

Curated by ChEMBL
LigandPNGBDBM4706((2R,3R,4S)-3-acetamido-4-hydroxy-2-[(1R,2R)-1,2,3-...)
Affinity DataKi:  1.23E+7nMAssay Description:Inhibition of Trypanosoma cruzi trans-SialidaseMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50520331(CHEMBL4445137)
Affinity DataIC50: <1nMAssay Description:Inhibition of human N-myristoyltransferase assessed as reduction in CoASH production by fluorogenic detection based assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50520335(CHEMBL4465173)
Affinity DataIC50: <1nMAssay Description:Inhibition of beta2 adrenoreceptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50132988(4-[3-(6-Bromo-pyridin-2-yl)-1H-pyrazol-4-yl]-quino...)
Affinity DataIC50:  1.20nMAssay Description:In vitro inhibition of transforming growth factor- beta dependent luciferase growth in mouse fibroblasts (NIH 3T3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50520336(CHEMBL4470042)
Affinity DataIC50:  2nMAssay Description:Inhibition of human PDE10A2 using cAMP substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDiscoidin domain-containing receptor 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataIC50:  2nMAssay Description:Inhibition of DDR2 (unknown origin) after 1 hr by time resolved fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHematopoietic prostaglandin D synthase(Homo sapiens (Human))TBA
LigandPNGBDBM50615811(CHEMBL5272869)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE3 cells assessed as reduction in PGD2 production using PGH2 as substrate by RapidFire...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
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