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Found 119 with Last Name = 'muller' and Initial = 'g'
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

LigandPNGBDBM8117(Hydroxyethylene Sulfone 17b | N-[(2S,3R,5S)-1-(3-b...)
Affinity DataKi:  45nM ΔG°:  -41.9kJ/mole IC50:  85nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

LigandPNGBDBM8123(Hydroxyethylene Sulfone 18a | N-((1S,2R,4S)-1-(3-b...)
Affinity DataKi:  370nM ΔG°:  -36.7kJ/mole IC50:  530nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

LigandPNGBDBM8124(Hydroxyethylene Sulfone 18b | N-((1S,2R,4S)-1-(3-b...)
Affinity DataKi:  540nM ΔG°:  -35.8kJ/mole IC50:  790nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

LigandPNGBDBM8118(Hydroxyethylene Sulfone 17b- | N-[(2R,3S,5R)-1-(3-...)
Affinity DataKi:  1.40E+3nM ΔG°:  -33.4kJ/mole IC50:  2.00E+3nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

LigandPNGBDBM8121((2R)-N-[(2S,3R,5S)-1-(3-bromophenyl)-7-(2,4-dichlo...)
Affinity DataKi:  2.90E+3nM ΔG°:  -31.6kJ/mole IC50:  4.20E+3nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

LigandPNGBDBM8120(2-bromo-N-[(2S,3R,5S)-1-(3-bromophenyl)-7-(2,4-dic...)
Affinity DataKi:  3.10E+3nM ΔG°:  -31.4kJ/mole IC50:  4.50E+3nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

LigandPNGBDBM8119(Hydroxyethylene Sulfone 17c | N-[(2S,3R,5S)-1-(3-b...)
Affinity DataKi:  7.00E+3nM ΔG°:  -29.4kJ/mole IC50:  1.00E+4nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

LigandPNGBDBM8122((2R)-N-[(2R,3S,5R)-1-(3-bromophenyl)-7-(2,4-dichlo...)
Affinity DataKi: >4.00E+4nM ΔG°: >-25.1kJ/mole IC50: >4.00E+4nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Philipps-Universitat Marburg

LigandPNGBDBM8116(Hydroxyethylene Sulfone 17a | N-[(2S,3R,5S)-1-(3-b...)
Affinity DataKi: >4.00E+4nM ΔG°: >-25.1kJ/mole IC50: >4.00E+4nMpH: 5.5 T: 2°CAssay Description:The inhibition assays were performed by mixing enzyme and fluorogenic substrate in the presence of inhibitor compounds. The hydrolysis of the substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484445(CHEMBL1916064)
Affinity DataIC50:  41nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484403(CHEMBL1916063)
Affinity DataIC50:  47nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484400(CHEMBL1916075)
Affinity DataIC50:  49nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484401(CHEMBL1916065)
Affinity DataIC50:  52nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484405(CHEMBL1915853)
Affinity DataIC50:  54nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA damage-binding protein 1/Protein cereblon(Homo sapiens (Human))
Celgene

LigandPNGBDBM65497(CC-220 (Compound 6) | US9694015, 6.4S)
Affinity DataIC50:  60nMpH: 7.0Assay Description:The 6XHis-tagged full length human CRBN bound to full length human DDB1 used in the assay was purified as described elsewhere with the exception that...More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484442(CHEMBL1916076)
Affinity DataIC50:  69nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484428(CHEMBL1916060)
Affinity DataIC50:  70nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484449(CHEMBL1916066)
Affinity DataIC50:  70nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484406(CHEMBL1915854)
Affinity DataIC50:  70nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484432(CHEMBL1916058)
Affinity DataIC50:  82nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484429(CHEMBL1915855)
Affinity DataIC50:  83nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484435(CHEMBL1916062)
Affinity DataIC50:  91nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
Sanofi

US Patent
LigandPNGBDBM141540(US8921404, 5)
Affinity DataIC50:  100nMpH: 7.0 T: 2°CAssay Description:To prepare the substrate, 25-50 uCi of [3H]trioleoylglycerol (in toluene), 6.8 umol of unlabeled trioleoylglycerol and 0.6 mg of phospholipids (phosp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
Sanofi

US Patent
LigandPNGBDBM141539(US8921404, 4)
Affinity DataIC50:  100nMpH: 7.0 T: 2°CAssay Description:To prepare the substrate, 25-50 uCi of [3H]trioleoylglycerol (in toluene), 6.8 umol of unlabeled trioleoylglycerol and 0.6 mg of phospholipids (phosp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
Sanofi

US Patent
LigandPNGBDBM141538(US8921404, 3)
Affinity DataIC50:  100nMpH: 7.0 T: 2°CAssay Description:To prepare the substrate, 25-50 uCi of [3H]trioleoylglycerol (in toluene), 6.8 umol of unlabeled trioleoylglycerol and 0.6 mg of phospholipids (phosp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484402(CHEMBL1916059)
Affinity DataIC50:  110nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
Sanofi

US Patent
LigandPNGBDBM141536(US8921404, 1)
Affinity DataIC50:  120nMpH: 7.0 T: 2°CAssay Description:To prepare the substrate, 25-50 uCi of [3H]trioleoylglycerol (in toluene), 6.8 umol of unlabeled trioleoylglycerol and 0.6 mg of phospholipids (phosp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
Sanofi

US Patent
LigandPNGBDBM141537(US8921404, 2)
Affinity DataIC50:  120nMpH: 7.0 T: 2°CAssay Description:To prepare the substrate, 25-50 uCi of [3H]trioleoylglycerol (in toluene), 6.8 umol of unlabeled trioleoylglycerol and 0.6 mg of phospholipids (phosp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484434(CHEMBL1916074)
Affinity DataIC50:  120nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484404(CHEMBL1916077)
Affinity DataIC50:  120nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50216304(CHEMBL313439)
Affinity DataIC50:  130nMAssay Description:Inhibition of PDE4 enzyme from U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484446(CHEMBL1915843)
Affinity DataIC50:  140nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484408(CHEMBL1915827)
Affinity DataIC50:  150nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484407(CHEMBL1916073)
Affinity DataIC50:  150nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484409(CHEMBL1915832)
Affinity DataIC50:  160nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484436(CHEMBL1915831)
Affinity DataIC50:  190nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484424(CHEMBL1916061)
Affinity DataIC50:  200nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50216301(CHEMBL88475)
Affinity DataIC50:  230nMAssay Description:Inhibition of PDE4 enzyme from U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
Sanofi

US Patent
LigandPNGBDBM141544(US8921404, 11)
Affinity DataIC50:  260nMpH: 7.0 T: 2°CAssay Description:To prepare the substrate, 25-50 uCi of [3H]trioleoylglycerol (in toluene), 6.8 umol of unlabeled trioleoylglycerol and 0.6 mg of phospholipids (phosp...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484433(3,3-Bis(3,4-Dimethoxyphenyl)Acrylonitrile | CHEMBL...)
Affinity DataIC50:  310nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50216299(CHEMBL315529)
Affinity DataIC50:  350nMAssay Description:Inhibition of PDE4 enzyme from U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484437(CHEMBL1915825)
Affinity DataIC50:  350nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484410(CHEMBL1916068)
Affinity DataIC50:  360nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484425(CHEMBL1916067)
Affinity DataIC50:  380nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTumor necrosis factor(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50052612(3-(5-Amino-1,3-dioxo-1,3-dihydro-isoindol-2-yl)-3-...)
Affinity DataIC50:  380nMAssay Description:Inhibition of TNF-alpha production in LPS stimulated human PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484411(CHEMBL1916072)
Affinity DataIC50:  400nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataIC50:  400nMAssay Description:Inhibition of phosphodiesterase 4 from U937 cellsMore data for this Ligand-Target Pair
TargetTumor necrosis factor(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50052602(3-(4-Amino-1,3-dioxo-1,3-dihydro-isoindol-2-yl)-3-...)
Affinity DataIC50:  450nMAssay Description:Inhibition of TNF-alpha production in LPS stimulated human PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM50484443(CHEMBL1916070)
Affinity DataIC50:  590nMAssay Description:Inhibition of human PDE4 expressed in U937 cells using [3H]cAMP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHormone-sensitive lipase(Rattus norvegicus (Rat))
Sanofi

US Patent
LigandPNGBDBM141543(US8921404, 10)
Affinity DataIC50:  670nMpH: 7.0 T: 2°CAssay Description:To prepare the substrate, 25-50 uCi of [3H]trioleoylglycerol (in toluene), 6.8 umol of unlabeled trioleoylglycerol and 0.6 mg of phospholipids (phosp...More data for this Ligand-Target Pair
In DepthDetails US Patent
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