Affinity DataEC50: 6.70nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.5nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 65nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 420nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.30nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 81nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.50E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.60nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 65nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 49nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 370nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 840nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 540nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 310nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.10E+3nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 99nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+3nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 96nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 760nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 78nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 290nMAssay Description:Agonist activity at rat GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Daiichi Sankyo
Curated by ChEMBL
Daiichi Sankyo
Curated by ChEMBL
Affinity DataEC50: 1.04E+4nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 330nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair