Affinity DataKi: 7.30E+3nMAssay Description:Inhibition of Influenza A virus (A/Indonesia/5/2005(H5N1)) X-31 recombinant neuraminidase using 2'-(4-methylumbelliferyl)-alpha-D-N-acetylneuraminic ...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of Influenza A virus (A/Sydney/5/97(H3N2)) recombinant neuraminidase using 2'-(4- methylumbelliferyl)-alpha-D-N-acetylneuraminic acid as s...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: >10nMAssay Description:Inhibition of human 11beta-HSD2More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of bovine platelet PDE5More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of Influenza A virus (A/Indonesia/5/2005(H5N1)) X-31 recombinant neuraminidase using 2'-(4-methylumbelliferyl)-alpha-D-N-acetylneuraminic ...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of human 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Yonsei University
Curated by ChEMBL
Yonsei University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human TACEMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Korea Basic Science Institute
Curated by ChEMBL
Korea Basic Science Institute
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of HA-EGFP tagged Plk1 polo-box domain (unknown origin) expressed in 293A cells assessed as inhibition of biotin-p-T78 binding after 1 hr ...More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Incheon National University
Curated by ChEMBL
Incheon National University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of mouse 11beta-HSD1More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of HDAC in HeLa cells by fluorescent activity assayMore data for this Ligand-Target Pair