TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 6.90nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membrane.More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 91nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 173nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 254nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York
Curated by ChEMBL
State University Of New York
Curated by ChEMBL
Affinity DataKi: 417nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.88E+3nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.08E+3nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.90E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.40E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.13E+5nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.17E+5nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.47E+5nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair