Compile Data Set for Download or QSAR
maximum 50k data
Found 63 with Last Name = 'natale' and Initial = 'nr'
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079458(2,6-Dimethyl-4-[3-methyl-5-(2-naphthalen-1-yl-ethy...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079458(2,6-Dimethyl-4-[3-methyl-5-(2-naphthalen-1-yl-ethy...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079463(4-{5-[2-(3-Bromo-phenyl)-ethyl]-3-phenyl-isoxazol-...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079463(4-{5-[2-(3-Bromo-phenyl)-ethyl]-3-phenyl-isoxazol-...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079459(4-[5-(2-Biphenyl-4-yl-ethyl)-3-methyl-isoxazol-4-y...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079464(2,6-Dimethyl-4-[3-methyl-5-(2-naphthalen-2-yl-ethy...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013025(2,6-Dimethyl-4-(5-methyl-3-phenyl-isoxazol-4-yl)-1...)
Affinity DataKi:  14nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079459(4-[5-(2-Biphenyl-4-yl-ethyl)-3-methyl-isoxazol-4-y...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079464(2,6-Dimethyl-4-[3-methyl-5-(2-naphthalen-2-yl-ethy...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013025(2,6-Dimethyl-4-(5-methyl-3-phenyl-isoxazol-4-yl)-1...)
Affinity DataKi:  22nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079462(2,6-Dimethyl-4-(3-methyl-5-phenethyl-isoxazol-4-yl...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079462(2,6-Dimethyl-4-(3-methyl-5-phenethyl-isoxazol-4-yl...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013022(4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...)
Affinity DataKi:  27nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013022(4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...)
Affinity DataKi:  29nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079460(4-{5-[2-(3-Methoxy-phenyl)-ethyl]-3-phenyl-isoxazo...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013022(4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...)
Affinity DataKi:  30nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50105838(FENOBAM)
Affinity DataKi:  32nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013022(4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...)
Affinity DataKi:  33nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50105838(FENOBAM)
Affinity DataKi:  33nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079460(4-{5-[2-(3-Methoxy-phenyl)-ethyl]-3-phenyl-isoxazo...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079465(4-[5-(2-Biphenyl-2-yl-ethyl)-3-methyl-isoxazol-4-y...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013021(4-(5-Ethyl-3-methyl-isoxazol-4-yl)-2,6-dimethyl-1,...)
Affinity DataKi:  52nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079461(2,6-Dimethyl-4-(5-phenethyl-3-phenyl-isoxazol-4-yl...)
Affinity DataKi:  55nMAssay Description:Displacement of [3H](+)-PN200-110 binding from calcium channels of rat cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013021(4-(5-Ethyl-3-methyl-isoxazol-4-yl)-2,6-dimethyl-1,...)
Affinity DataKi:  63nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079461(2,6-Dimethyl-4-(5-phenethyl-3-phenyl-isoxazol-4-yl...)
Affinity DataKi:  73nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013026(2,6-Dimethyl-4-(5-pentyl-3-phenyl-isoxazol-4-yl)-1...)
Affinity DataKi:  78nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013026(2,6-Dimethyl-4-(5-pentyl-3-phenyl-isoxazol-4-yl)-1...)
Affinity DataKi:  79nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50079465(4-[5-(2-Biphenyl-2-yl-ethyl)-3-methyl-isoxazol-4-y...)
Affinity DataKi:  91nMAssay Description:Displacement of [3H](+)-PN200-110 binding to calcium channels in guinea pig cardiac membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013024(4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...)
Affinity DataKi:  122nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013024(4-(3,5-Dimethyl-isoxazol-4-yl)-2,6-dimethyl-1,4-di...)
Affinity DataKi:  173nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1F/alpha-1S(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013023(4-(5-Isopropyl-3-phenyl-isoxazol-4-yl)-2,6-dimethy...)
Affinity DataKi:  254nMAssay Description:Inhibition of [3H]PN-200110 binding to Calcium channel in guinea pig ileum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50013023(4-(5-Isopropyl-3-phenyl-isoxazol-4-yl)-2,6-dimethy...)
Affinity DataKi:  417nMAssay Description:Inhibition of [3H]-PN-200110 binding to Calcium channel in guinea pig heart membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50450061(CHEMBL4166199)
Affinity DataKi:  1.88E+3nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50450078(CHEMBL4167825)
Affinity DataKi:  3.08E+3nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50450074(CHEMBL4171187)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50450059(CHEMBL4160584)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50450076(CHEMBL4163974)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50450077(CHEMBL4164391)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50450075(CHEMBL4174628)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50450060(CHEMBL4172276)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of MPEP from mGluR5 (unknown origin) after 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378670(CHEMBL600474)
Affinity DataKi:  5.20E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50109609((2R)-2-amino-3-mercaptopropanoic acid | (2R)-2-ami...)
Affinity DataKi:  5.90E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378666(CHEMBL601837)
Affinity DataKi:  6.00E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378667(CHEMBL604574)
Affinity DataKi:  6.40E+4nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378668(CHEMBL606915)
Affinity DataKi:  1.13E+5nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378669(CHEMBL591770)
Affinity DataKi:  1.17E+5nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50378665(CHEMBL590556)
Affinity DataKi:  1.47E+5nMAssay Description:Competitive inhibition of [3H]L-glutamate uptake at amino acid transport system xc- in human SNB19 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242247(CHEMBL4074268)
Affinity DataIC50:  510nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242253(CHEMBL4092304)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Montana

Curated by ChEMBL
LigandPNGBDBM50242254(CHEMBL4104354)
Affinity DataIC50:  1.39E+3nMAssay Description:Inhibition of MDR-1 in human Caco-2 cells after 30 mins by calcein-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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