Compile Data Set for Download or QSAR
maximum 50k data
Found 61 with Last Name = 'nazareno' and Initial = 'dv'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50095105(4-{2-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenyl]-[1,...)
Affinity DataKi:  0.0100nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103771((4-{2-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-[1,3]...)
Affinity DataKi:  0.140nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103774((5-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  0.200nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103772((5,7-Difluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy...)
Affinity DataKi:  0.230nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103767((5,8-Difluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy...)
Affinity DataKi:  0.290nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103773((4-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  0.510nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103768((5-Bromo-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-benz...)
Affinity DataKi:  0.510nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103087(CHEMBL305026 | [4-((R)-4-{(S)-1-[4-(Benzo[1,3]diox...)
Affinity DataKi:  0.800nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103775((6-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  0.810nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103769((8-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  0.990nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103078(CHEMBL67563 | [4-(4-{(S)-1-[4-(Benzo[1,3]dioxole-5...)
Affinity DataKi:  1nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103770((7-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  1.20nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103776((6-Chloro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  1.40nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104946((2,4-Dimethyl-pyridin-3-yl)-(4-methyl-4-{(S)-3-met...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity at C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104950((2,6-Dimethyl-phenyl)-(4-{(S)-4-[(S)-1-(4-methanes...)
Affinity DataKi:  3nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104958((2-Amino-6-chloro-phenyl)-(4-{(S)-4-[(S)-1-(4-meth...)
Affinity DataKi:  5nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104953((2-Amino-6-chloro-phenyl)-(4-{(S)-4-[(S)-1-(4-iodo...)
Affinity DataKi:  5nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104955((2-Amino-6-chloro-phenyl)-(4-methyl-4-{(S)-3-methy...)
Affinity DataKi:  5nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104952((2,6-Dimethyl-phenyl)-(4-{(S)-4-[(S)-1-(4-iodo-phe...)
Affinity DataKi:  5nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104944((2-Hydroxy-6-methyl-phenyl)-(4-methyl-4-{(S)-3-met...)
Affinity DataKi:  5nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104954((2,6-Dimethyl-phenyl)-(4-methyl-4-{(S)-3-methyl-4-...)
Affinity DataKi:  7nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104956((2,4-Dimethyl-1-oxy-pyridin-3-yl)-(4-methyl-4-{(S)...)
Affinity DataKi:  7nMAssay Description:Binding affinity at C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104949((2,6-Dimethyl-phenyl)-{4-[(S)-4-(4-iodo-benzyl)-3-...)
Affinity DataKi:  8nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104951((2-Hydroxy-6-methyl-phenyl)-(4-{(S)-4-[(S)-1-(4-io...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104959((2-Hydroxy-6-methyl-phenyl)-(4-{(S)-4-[(S)-1-(4-me...)
Affinity DataKi:  15nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103083((4-{(S)-4-[(S)-1-(4-Benzo[1,3]dioxol-5-ylmethyl-ph...)
Affinity DataKi:  18nMAssay Description:Inhibition of [125I]-labeled RANTES binding to C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104957((2,6-Dimethyl-phenyl)-(4-{(S)-4-[(S)-1-(4-iodo-phe...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104947((4-{4-[1-(4-Bromo-phenyl)-ethyl]-3-methyl-piperazi...)
Affinity DataKi:  23nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103088(CHEMBL70010 | [4-((S)-4-{(S)-1-[4-(Benzo[1,3]dioxo...)
Affinity DataKi:  28nMAssay Description:Inhibition of [125I]-labeled RANTES binding to C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104961((2,6-Dimethyl-phenyl)-{4-[(S)-4-(4-iodo-benzyl)-3-...)
Affinity DataKi:  30nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103091((4-{4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-benzyl]-pi...)
Affinity DataKi:  31nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103080((2-Amino-6-methyl-phenyl)-[4-((S)-4-{(S)-1-[4-(ben...)
Affinity DataKi:  31nMAssay Description:Ability of the compound to inhibit [125I]-labeled RANTES binding to C-C chemokine receptor type 5 expressed in membrane preparation of CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103085((2-Amino-6-chloro-phenyl)-[4-((S)-4-{(S)-1-[4-(ben...)
Affinity DataKi:  32nMAssay Description:Inhibition of [125I]-labeled RANTES binding to C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103777(4-{2-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-[1,3]d...)
Affinity DataKi:  33nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103090((4-{(S)-4-[(S)-1-(4-Benzo[1,3]dioxol-5-ylmethyl-ph...)
Affinity DataKi:  35nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103084(CHEMBL66623 | {4-[(S)-4-(4-Benzo[1,3]dioxol-5-ylme...)
Affinity DataKi: >40nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103089((4-{(S)-4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-benzyl...)
Affinity DataKi: >40nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103084(CHEMBL66623 | {4-[(S)-4-(4-Benzo[1,3]dioxol-5-ylme...)
Affinity DataKi:  44nMAssay Description:Inhibition of [125I]-labeled RANTES binding to C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103086(CHEMBL413972 | [4-((S)-4-{(S)-1-[4-(3-Chloro-benzy...)
Affinity DataKi:  45nMAssay Description:Inhibition of [125I]-labeled RANTES binding to C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103079(CHEMBL303503 | [4-((S)-4-{(S)-1-[4-(Benzo[1,3]diox...)
Affinity DataKi:  49nMAssay Description:Inhibition of [125I]-labeled RANTES binding to C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104960((2,6-Dimethyl-phenyl)-{4-[4-(4-iodo-benzyl)-pipera...)
Affinity DataKi:  62nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103089((4-{(S)-4-[4-(Benzo[1,3]dioxole-5-sulfonyl)-benzyl...)
Affinity DataKi:  74nMAssay Description:Inhibition of [125I]-labeled RANTES binding to C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103085((2-Amino-6-chloro-phenyl)-[4-((S)-4-{(S)-1-[4-(ben...)
Affinity DataKi:  100nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103080((2-Amino-6-methyl-phenyl)-[4-((S)-4-{(S)-1-[4-(ben...)
Affinity DataKi:  100nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103082(CHEMBL67281 | [4-((S)-4-{(S)-1-[4-(Benzo[1,3]dioxo...)
Affinity DataKi:  230nMAssay Description:Inhibition of [125I]-labeled RANTES binding to C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104956((2,4-Dimethyl-1-oxy-pyridin-3-yl)-(4-methyl-4-{(S)...)
Affinity DataKi:  250nMAssay Description:Binding affinity against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103079(CHEMBL303503 | [4-((S)-4-{(S)-1-[4-(Benzo[1,3]diox...)
Affinity DataKi:  270nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104945((2,6-Dimethyl-phenyl)-{4-[3-methyl-4-(1-phenyl-eth...)
Affinity DataKi:  275nMAssay Description:Binding affinity towards C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103082(CHEMBL67281 | [4-((S)-4-{(S)-1-[4-(Benzo[1,3]dioxo...)
Affinity DataKi:  352nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103081(CHEMBL63757 | {4-[4-(4-Benzo[1,3]dioxol-5-ylmethyl...)
Affinity DataKi:  352nMAssay Description:Inhibition of [125I]-labeled RANTES binding to C-C chemokine receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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