TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of flag-tagged HDAC3More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of flag-tagged HDAC4 by Biomol assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of flag-tagged HDAC4More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of flag-tagged HDAC4More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of flag-tagged HDAC4 by Biomol assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of flag-tagged HDAC4 by pull-down assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of HDAC4 catalytic domain expressed in HEK293 cells by Biomol assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of flag-tagged HDAC3More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of flag-tagged HDAC4 expressed in HEK293 cells by Biomol assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 3.60nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of flag-tagged HDAC4 by pull-down assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMpH: 7.5 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMT: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 9.70nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 10nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMT: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 24nMpH: 7.5 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 33nMT: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 43nMT: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 46nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 57nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Inhibition of flag-tagged HDAC4 by Biomol assayMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 120nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 130nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 152nMAssay Description:Inhibition of flag-tagged HDAC4 by pull-down assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMpH: 7.5 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 400nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human CKIdeltaMore data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 420nMT: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of flag-tagged HDAC4 by pull-down assayMore data for this Ligand-Target Pair
Affinity DataIC50: 540nMpH: 7.5 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 610nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human CKIalphaMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human CKIalphaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMpH: 8.0 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human CKIdeltaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMT: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of flag-tagged HDAC4 by Biomol assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMpH: 7.5 T: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMT: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare
Curated by ChEMBL
Affinity DataIC50: 8.70E+3nMT: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of human RSK2More data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of human RSK2More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Istituto Di Ricerche Di Biologia Molecolare &Quot;P. Angeletti
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CK2More data for this Ligand-Target Pair