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Found 24 with Last Name = 'negi' and Initial = 'as'
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM19461(α-CA inhibitor, 5 | 5,7-dihydroxy-2-(4-hydrox...)
Affinity DataKi:  0.00110nM IC50:  1.00E+3nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92556(Neoflavonoid, 8)
Affinity DataKi:  0.00182nM IC50:  1.21E+4nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92555(Neoflavonoid, 7)
Affinity DataKi:  0.00216nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92557(Neoflavonoid, 9)
Affinity DataKi:  0.00256nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92559(Neoflavonoid, 11)
Affinity DataKi:  0.00425nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92560(Neoflavonoid, 19)
Affinity DataKi:  0.00597nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92558(Neoflavonoid, 10)
Affinity DataKi:  0.00838nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Central Institute of Medicinal and Aromatic Plants

LigandPNGBDBM92561(Neoflavonoid, 20)
Affinity DataKi:  0.0118nMAssay Description:Inhibition assay using aromatase enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM912((3S,4S)-3-hydroxy-4-[(2S)-2-[(3S,4S)-3-hydroxy-6-m...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM50189981(2-[1-(3,4,5-trimethoxybenzoyl)naphthalen-2-yloxy]e...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM50189983(CHEMBL214974 | N-butyl-4-(1-(3,4,5-trimethoxybenzo...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM50189976(CHEMBL212492 | N-(4-methoxyphenyl)-4-(1-(3,4,5-tri...)
Affinity DataIC50:  4.71E+3nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM50189980(CHEMBL213373 | N-octyl-2-(1-(3,4,5-trimethoxybenzo...)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM50189985(4-[1-(3,4,5-trimethoxybenzoyl)naphthalen-2-yloxy]-...)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Csir-Central Institute Of Medicinal And Aromatic Plants (Csir-Cimap)

Curated by ChEMBL
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)
Affinity DataIC50:  3.77E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase supercoiling activity using relaxed pBR322 as substrate after 30 mins by agarose gel electrophore...More data for this Ligand-Target Pair
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Csir-Central Institute Of Medicinal And Aromatic Plants (Csir-Cimap)

Curated by ChEMBL
LigandPNGBDBM50463548(CHEMBL4239753)
Affinity DataIC50:  8.57E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase supercoiling activity using relaxed pBR322 as substrate after 30 mins by agarose gel electrophore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM50189984(CHEMBL378015 | N-phenyl-2-(1-(3,4,5-trimethoxybenz...)
Affinity DataIC50:  2.32E+5nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Csir-Central Institute Of Medicinal And Aromatic Plants (Csir-Cimap)

Curated by ChEMBL
LigandPNGBDBM50463549(CHEMBL4237298)
Affinity DataIC50:  2.94E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase supercoiling activity using relaxed pBR322 as substrate after 30 mins by agarose gel electrophore...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Csir-Central Institute Of Medicinal And Aromatic Plants (Csir-Cimap)

Curated by ChEMBL
LigandPNGBDBM50463550(CHEMBL4251156)
Affinity DataIC50:  3.58E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase supercoiling activity using relaxed pBR322 as substrate after 30 mins by agarose gel electrophore...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Csir-Central Institute Of Medicinal And Aromatic Plants (Csir-Cimap)

Curated by ChEMBL
LigandPNGBDBM50463551(CHEMBL4243541)
Affinity DataIC50:  3.80E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis DNA gyrase supercoiling activity using relaxed pBR322 as substrate after 30 mins by agarose gel electrophore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM50189979(CHEMBL378329 | N-phenyl-4-(1-(3,4,5-trimethoxybenz...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM50189978(CHEMBL377142 | N-(4-methoxyphenyl)-2-(1-(3,4,5-tri...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM50189977(4-(1-(3,4,5-trimethoxybenzoyl)naphthalen-2-yloxy)b...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Institute Of Medicinal And Aromatic Plants

Curated by ChEMBL
LigandPNGBDBM50189982(2-[1-(3,4,5-trimethoxybenzoyl)naphthalene-2-yloxy]...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed