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Found 394 with Last Name = 'nishimura' and Initial = 'y'
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50318885(CHEMBL525610 | teriparatide)
Affinity DataIC50:  0.0800nMAssay Description:Displacement of 125I-PTH (1 to 15 residues) from human PTHR1 expressed in African green monkey COS7 cell membranes at 300 uM after 90 mins by gamma c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445769(CHEMBL3104615)
Affinity DataIC50:  0.125nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441476(CHEMBL2436575)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441467(CHEMBL2436573)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441481(CHEMBL2436579)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50192809(CHEMBL3941914)
Affinity DataIC50:  0.220nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441483(CHEMBL2436591)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441469(CHEMBL2436586)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441470(CHEMBL2436574)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441474(CHEMBL2436563)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50192811(CHEMBL3971502)
Affinity DataIC50:  0.300nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50192807(CHEMBL3984947)
Affinity DataIC50:  0.360nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441486(CHEMBL2436593)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441472(CHEMBL2436578)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441468(CHEMBL2436564)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50192809(CHEMBL3941914)
Affinity DataIC50:  0.400nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of hypotonicity-induced activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445752(CHEMBL3104441)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441482(CHEMBL2436577)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441492(CHEMBL2436580)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445751(CHEMBL3104442)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441484(CHEMBL2436587)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50192804(CHEMBL3933401)
Affinity DataIC50:  0.570nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441479(CHEMBL2436590)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441475(CHEMBL2436589)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445760(CHEMBL3104432)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445758(CHEMBL3104435)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445753(CHEMBL3104440)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50276045((R)-3-Amino-4-(5-chloro-2-fluoro-phenyl)-N-{4-[6-(...)
Affinity DataIC50:  0.640nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441471(CHEMBL2436572)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445770(CHEMBL3104444)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441478(CHEMBL2436584)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445750(CHEMBL3104443)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50276047((R)-3-Amino-N-{4-[6-(2-morpholin-4-yl-ethoxy)-benz...)
Affinity DataIC50:  0.790nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441488(CHEMBL2436592)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441487(CHEMBL2436576)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445763(CHEMBL3104622)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445757(CHEMBL3104436)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441480(CHEMBL2436581)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50192820(CHEMBL3950646)
Affinity DataIC50:  0.900nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50192808(CHEMBL3915150)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50276001((R)-3-Amino-N-{4-[6-(2-methoxy-ethoxy)-benzothiazo...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human Caco2 cells-derived DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445764(CHEMBL3104621)
Affinity DataIC50:  1nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441461(CHEMBL2436568)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50192779(CHEMBL3957347)
Affinity DataIC50:  1.10nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445768(CHEMBL3102876)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445759(CHEMBL3104433)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445765(CHEMBL3104620)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50441462(CHEMBL2436585)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human recombinant sEH using cyano(6-methoxy-naphthalen-2-yl)methyl trans-[(3-phenyloxiran-2-yl)methyl]carbonate after 20 to 45 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50182869(CHEMBL439521 | N-((S)-2-amino-3-((S)-1-((S)-1-((2S...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human recombinant BACE1 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50445767(CHEMBL3104617)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human recombinant sEH expressed in baculovirus infected insect Sf9 cells using cyano(6-methoxynaphthalen-2-yl)methyl trans-[(3-phenylox...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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