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Found 1494 with Last Name = 'norris' and Initial = 'jl'
TargetMelanoma-associated antigen 4(Homo sapiens)
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50605667(CHEMBL5187815)
Affinity DataIC50: <1nMAssay Description:Inhibition of Eu-W1024 streptavidin-labeled MAGEA4 (unknown origin) expressed in Escherichia coli BL21-(DE3) incubated for 30 to 60 mins by LANCE TR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMelanoma-associated antigen 4(Homo sapiens)
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50605668(CHEMBL5199001)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of Eu-W1024 streptavidin-labeled MAGEA4 (unknown origin) expressed in Escherichia coli BL21-(DE3) incubated for 30 to 60 mins by LANCE TR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMelanoma-associated antigen 4(Homo sapiens)
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50605666(CHEMBL5188210)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Eu-W1024 streptavidin-labeled MAGEA4 (unknown origin) expressed in Escherichia coli BL21-(DE3) incubated for 30 to 60 mins by LANCE TR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMelanoma-associated antigen 4(Homo sapiens)
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50605669(CHEMBL5208958)
Affinity DataIC50:  11nMAssay Description:Inhibition of Eu-W1024 streptavidin-labeled MAGEA4 (unknown origin) expressed in Escherichia coli BL21-(DE3) incubated for 30 to 60 mins by LANCE TR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMelanoma-associated antigen 4(Homo sapiens)
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50605670(CHEMBL5182108)
Affinity DataIC50:  14nMAssay Description:Inhibition of Eu-W1024 streptavidin-labeled MAGEA4 (unknown origin) expressed in Escherichia coli BL21-(DE3) incubated for 30 to 60 mins by LANCE TR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50323813(7-(2-(2-(Dimethylamino)ethoxy)ethoxy)-6-methoxy-2-...)
Affinity DataIC50:  15nMAssay Description:Activity at methyl transferase activity GLP by enzyme coupled S-adenocylehomocystein detection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50323813(7-(2-(2-(Dimethylamino)ethoxy)ethoxy)-6-methoxy-2-...)
Affinity DataIC50:  23nMAssay Description:Activity at methyl transferase activity GLP by chemiluminescence based oxygen tunneling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440614(CHEMBL2426364)
Affinity DataIC50:  24nMAssay Description:Inhibition of His-tagged L3MBTL3 (unknown origin) using H4K20Me2 as substrate incubated for 30 mins at room temperature followed by incubation under ...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50300028(CHEMBL569864 | N-(1-benzylpiperidin-4-yl)-6,7-dime...)
Affinity DataIC50:  27nMAssay Description:Activity at methyl transferase activity GLP by chemiluminescence based oxygen tunneling assayMore data for this Ligand-Target Pair
TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194448(CHEMBL3972289)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50300028(CHEMBL569864 | N-(1-benzylpiperidin-4-yl)-6,7-dime...)
Affinity DataIC50:  34nMAssay Description:Activity at methyl transferase activity GLP by enzyme coupled S-adenocylehomocystein detection assayMore data for this Ligand-Target Pair
TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194466(CHEMBL3958557)
Affinity DataIC50:  35nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194475(CHEMBL3889586)
Affinity DataIC50:  35nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194259(CHEMBL3939958)
Affinity DataIC50:  37nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50496581(CHEMBL3134130)
Affinity DataIC50:  37nMAssay Description:Inhibition of His-tagged L3MBTL3 (unknown origin) using H4K20Me2 as substrate incubated for 30 mins at room temperature followed by incubation under ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440613(CHEMBL2426365)
Affinity DataIC50:  39nMAssay Description:Inhibition of L3MBTL3 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440563(CHEMBL2426360)
Affinity DataIC50:  43nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194476(CHEMBL3942693)
Affinity DataIC50:  47nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50496591(CHEMBL3134144)
Affinity DataIC50:  48nMAssay Description:Inhibition of His-tagged L3MBTL3 (unknown origin) using H4K20Me2 as substrate incubated for 30 mins at room temperature followed by incubation under ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440603(CHEMBL2426498)
Affinity DataIC50:  48nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440612(CHEMBL2426366)
Affinity DataIC50:  48nMAssay Description:Inhibition of L3MBTL3 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440614(CHEMBL2426364)
Affinity DataIC50:  49nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440613(CHEMBL2426365)
Affinity DataIC50:  50nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50300041(7-(3-(dimethylamino)propoxy)-6-methoxy-2-(4-methyl...)
Affinity DataIC50:  50nMAssay Description:Activity at methyl transferase activity GLP by enzyme coupled S-adenocylehomocystein detection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440612(CHEMBL2426366)
Affinity DataIC50:  51nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440611(CHEMBL2426367)
Affinity DataIC50:  53nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194477(CHEMBL3916023)
Affinity DataIC50:  56nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50300041(7-(3-(dimethylamino)propoxy)-6-methoxy-2-(4-methyl...)
Affinity DataIC50:  58nMAssay Description:Activity at methyl transferase activity GLP by chemiluminescence based oxygen tunneling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440611(CHEMBL2426367)
Affinity DataIC50:  58nMAssay Description:Inhibition of L3MBTL3 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50496584(CHEMBL3134146)
Affinity DataIC50:  59nMAssay Description:Inhibition of His-tagged L3MBTL3 (unknown origin) using H4K20Me2 as substrate incubated for 30 mins at room temperature followed by incubation under ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440610(CHEMBL2426368)
Affinity DataIC50:  61nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194258(CHEMBL3934881)
Affinity DataIC50:  61nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440569(CHEMBL2424678)
Affinity DataIC50:  61nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50496593(CHEMBL3134131)
Affinity DataIC50:  62nMAssay Description:Inhibition of His-tagged L3MBTL3 (unknown origin) using H4K20Me2 as substrate incubated for 30 mins at room temperature followed by incubation under ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetE3 SUMO-protein ligase CBX4(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194448(CHEMBL3972289)
Affinity DataIC50:  62nMAssay Description:Antagonist activity at recombinant human N-terminal His-tagged CBX4 chromodomain (8 to 65 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194458(CHEMBL3987134)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440614(CHEMBL2426364)
Affinity DataIC50:  64nMAssay Description:Inhibition of L3MBTL3 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440610(CHEMBL2426368)
Affinity DataIC50:  66nMAssay Description:Inhibition of L3MBTL3 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440560(CHEMBL2426363)
Affinity DataIC50:  68nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanoma-associated antigen 4(Homo sapiens)
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50605672(CHEMBL5197762)
Affinity DataIC50:  68nMAssay Description:Inhibition of Eu-W1024 streptavidin-labeled MAGEA4 (unknown origin) expressed in Escherichia coli BL21-(DE3) incubated for 30 to 60 mins by LANCE TR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50496596(CHEMBL3134134)
Affinity DataIC50:  70nMAssay Description:Inhibition of His-tagged L3MBTL3 (unknown origin) using H4K20Me2 as substrate incubated for 30 mins at room temperature followed by incubation under ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440603(CHEMBL2426498)
Affinity DataIC50:  71nMAssay Description:Inhibition of L3MBTL3 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440563(CHEMBL2426360)
Affinity DataIC50:  72nMAssay Description:Inhibition of L3MBTL3 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440585(CHEMBL2426496)
Affinity DataIC50:  74nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50440568(CHEMBL2426476)
Affinity DataIC50:  74nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 SUMO-protein ligase CBX4(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194475(CHEMBL3889586)
Affinity DataIC50:  75nMAssay Description:Antagonist activity at recombinant human N-terminal His-tagged CBX4 chromodomain (8 to 65 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromodomain Y-like protein 2(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194458(CHEMBL3987134)
Affinity DataIC50:  75nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CDYL2 chromodomain (1 to 75 residues) expressed in Escherichia coli Rosetta BL21(DE3)p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 7(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194457(CHEMBL3969494)
Affinity DataIC50:  75nMAssay Description:Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 SUMO-protein ligase CBX4(Homo sapiens (Human))
University Of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50194466(CHEMBL3958557)
Affinity DataIC50:  75nMAssay Description:Antagonist activity at recombinant human N-terminal His-tagged CBX4 chromodomain (8 to 65 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50496589(CHEMBL3134126)
Affinity DataIC50:  80nMAssay Description:Inhibition of His-tagged L3MBTL3 (unknown origin) using H4K20Me2 as substrate incubated for 30 mins at room temperature followed by incubation under ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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