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Found 323 with Last Name = 'o''neill' and Initial = 'ab'
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287851((S)-2-(3-Fluoro-phenoxymethyl)-azetidine | CHEMBL3...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  3.80nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287814((S)-2-(3-Fluoro-phenoxymethyl)-1-methyl-pyrrolidin...)
Affinity DataKi:  5nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  8.70nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118703(CHEMBL109783 | N-[5-(4,5-Dihydro-1H-imidazol-2-yl)...)
Affinity DataKi:  12nMAssay Description:Binding affinity towards rat submaxillary gland Alpha-1 adrenergic receptor; value ranges from (0.009 - 0.015)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118703(CHEMBL109783 | N-[5-(4,5-Dihydro-1H-imidazol-2-yl)...)
Affinity DataKi:  12nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287829((R)-2-(3-Fluoro-phenoxymethyl)-pyrrolidine | CHEMB...)
Affinity DataKi:  13nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287821((S)-2-(3-Fluoro-phenoxymethyl)-1-methyl-azetidine ...)
Affinity DataKi:  14nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287812((S)-2-(3-Fluoro-phenoxymethyl)-pyrrolidine | CHEMB...)
Affinity DataKi:  14nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287838((S)-2-(3,4-Difluoro-phenoxymethyl)-pyrrolidine | C...)
Affinity DataKi:  17nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287816((S)-2-(3,5-Difluoro-phenoxymethyl)-pyrrolidine | C...)
Affinity DataKi:  18nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287834(3-((S)-1-Pyrrolidin-2-ylmethoxy)-benzonitrile | CH...)
Affinity DataKi:  18nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287848((S)-2-(3,4-Difluoro-phenoxymethyl)-1-methyl-pyrrol...)
Affinity DataKi:  18nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287849((S)-2-(3,5-Difluoro-phenoxymethyl)-1-methyl-pyrrol...)
Affinity DataKi:  19nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474632(CHEMBL327116)
Affinity DataKi:  22nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474660(CHEMBL111771)
Affinity DataKi:  22nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474632(CHEMBL327116)
Affinity DataKi:  23nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  31nMAssay Description:In vitro binding affinity towards alpha-1D adrenergic receptor of rat clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118703(CHEMBL109783 | N-[5-(4,5-Dihydro-1H-imidazol-2-yl)...)
Affinity DataKi:  33nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataKi:  36nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287852((S)-2-(3-Chloro-phenoxymethyl)-1-methyl-pyrrolidin...)
Affinity DataKi:  37nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287824((S)-1-Methyl-2-phenoxymethyl-pyrrolidine | CHEMBL7...)
Affinity DataKi:  42nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataKi:  45nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474631(CHEMBL323004)
Affinity DataKi:  46nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474633(CHEMBL111496)
Affinity DataKi:  47nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataKi:  48nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataKi:  49nMAssay Description:In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287820(3-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-benzonitri...)
Affinity DataKi:  51nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287843((S)-2-Phenoxymethyl-azetidine | CHEMBL72031)
Affinity DataKi:  52nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287825((S)-2-(2,3-Difluoro-phenoxymethyl)-1-methyl-pyrrol...)
Affinity DataKi:  69nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataKi:  72nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287846((S)-2-(2,3-Difluoro-phenoxymethyl)-pyrrolidine | C...)
Affinity DataKi:  77nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287854((R)-2-(3-Fluoro-phenoxymethyl)-1-methyl-pyrrolidin...)
Affinity DataKi:  78nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474642(CHEMBL110975)
Affinity DataKi:  83nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474638(CHEMBL111463)
Affinity DataKi:  85nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474637(CHEMBL2111710)
Affinity DataKi:  91nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474660(CHEMBL111771)
Affinity DataKi:  98nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474644(CHEMBL112814)
Affinity DataKi:  100nMAssay Description:In vitro binding affinity towards alpha-1D adrenergic receptor of rat clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287842((S)-1-Methyl-2-phenoxymethyl-azetidine | CHEMBL754...)
Affinity DataKi:  101nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474671(CHEMBL111554)
Affinity DataKi:  105nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287830((R)-2-Phenoxymethyl-pyrrolidine | CHEMBL73784)
Affinity DataKi:  107nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287844((S)-2-(3,4-Dichloro-phenoxymethyl)-1-methyl-pyrrol...)
Affinity DataKi:  112nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(CALF)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  115nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of bovine clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474666(CHEMBL321644)
Affinity DataKi:  123nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474643(CHEMBL111734)
Affinity DataKi:  129nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474633(CHEMBL111496)
Affinity DataKi:  132nMAssay Description:In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  135nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287855(3-((S)-1-Pyrrolidin-2-ylmethoxy)-benzamide | CHEMB...)
Affinity DataKi:  136nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(CALF)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataKi:  138nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of bovine clone in radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  140nMAssay Description:Binding affinity towards rat submaxillary gland Alpha-1 adrenergic receptor ; value ranges from (0.12 - 0.15)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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