Affinity DataKi: 0.320nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.850nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding of Adenosine A2 receptor in whole rat brain membrane using [3H]CHA as a RadioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding of Adenosine A2 receptor in whole rat brain membrane using [3H]CHA as a RadioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]AMPA from homomeric recombinant GluA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding of Adenosine A2 receptor in whole rat brain membrane using [3H]CHA as a RadioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding of Adenosine A2 receptor in whole rat brain membrane using [3H]CHA as a RadioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding of Adenosine A2 receptor in whole rat brain membrane using [3H]CHA as a RadioligandMore data for this Ligand-Target Pair
Affinity DataKi: 23.2nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 25.3nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 32.6nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 33.5nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 49.4nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
Eli Lilly
Curated by PDSP Ki Database
Eli Lilly
Curated by PDSP Ki Database
Affinity DataKi: 60.7nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 64.3nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 73.8nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 94.3nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 94.6nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 96nMAssay Description:Inhibition of [3H]-CHA binding to Adenosine A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding of Adenosine A2 receptor in whole rat brain membrane using [3H]CHA as a RadioligandMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Inhibition of [3H]-CHA binding to rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 136nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 157nMAssay Description:Binding of Adenosine A2 receptor in whole rat brain membrane using [3H]CHA as a RadioligandMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 161nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 164nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
Affinity DataKi: 175nMAssay Description:Binding affinity towards adenosine A1 receptor was determined using radioligand [3H]-CHA in whole rat brain membranes at 25 degree CMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of [3H]-AMPA binding to human GluR2 receptors expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Ability to displace binding of [3H]AMPA to recombinant human Ionotropic glutamate receptor AMPA 2More data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Inhibition of [3H]-CHA binding to Adenosine A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Displacement of Bodipy-labelled cyclopamine from Smo expressed in COS-1 cells in presence of 2% FBS after 4 to 6 hrs by FACS flow cytometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Binding of Adenosine A2 receptor in whole rat brain membrane using [3H]CHA as a RadioligandMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair