Affinity DataKi: 3nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Laboratoire De Chimie ThéRapeutique Associé
Curated by ChEMBL
Laboratoire De Chimie ThéRapeutique Associé
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Binding affinity towards Tachykinin receptor 1 expressed in CHO cells using [3H]-[Pro9]-SP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of HIV1 protease dimerization expressed in Escherichia coli Rosetta(DE3) using DABCYL-gamma-abu-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-EDANS as s...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Inhibition of HIV1 protease dimerization expressed in Escherichia coli Rosetta(DE3) using DABCYL-gamma-abu-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-EDANS as s...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of dimerization of HIV1 protease 150V mutantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Laboratoire De Chimie ThéRapeutique Associé
Curated by ChEMBL
Laboratoire De Chimie ThéRapeutique Associé
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Binding affinity towards Tachykinin receptor 1 expressed in CHO cells using [3H]-[Pro9]-SP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition of HIV1 protease dimerization expressed in Escherichia coli Rosetta(DE3) using DABCYL-gamma-abu-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-EDANS as s...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of dimerization of HIV1 protease ANAM-11 mutantMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of wild type HIV1 protease dimerizationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Inhibition of dimerization of HIV1 protease V82A mutantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibition of wild type HIV1 protease dimerizationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 488nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of dimerization of HIV1 protease G48V/L90M mutantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of dimerization of HIV1 protease D30N mutantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Inhibition of HIV1 protease dimerization expressed in Escherichia coli Rosetta(DE3) using DABCYL-gamma-abu-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-EDANS as s...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University
Curated by ChEMBL
Paris-Sud University
Curated by ChEMBL
Affinity DataKi: 560nMAssay Description:Inhibition of dimerization of HIV1 proteaseMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Laboratoire De Chimie ThéRapeutique Associé
Curated by ChEMBL
Laboratoire De Chimie ThéRapeutique Associé
Curated by ChEMBL
Affinity DataKi: 620nMAssay Description:Binding affinity towards Tachykinin receptor 1 expressed in CHO cells using [3H]-[Pro9]-SP as radioligandMore data for this Ligand-Target Pair