TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 380nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 510nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 580nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 620nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 720nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 740nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 770nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 820nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 840nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 850nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 930nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 930nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 3.16E+3nMAssay Description:Displacement of [3H]-dofetilide from human ERG channel expressed in HEK293 by scintillation countingMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataKi: 5.30E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of maximum response evoked by cAMP on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 166nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development
Curated by ChEMBL
Research And Development
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 309nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 355nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Antagonist activity at human recombinant GnRHR expressed in CHOK1 cells assessed as reduction in luminescence signal by luciferase reporter gene assa...More data for this Ligand-Target Pair