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Found 723 with Last Name = 'oyama' and Initial = 'm'
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317865(2-(2-(4-tert-Butylphenylthio)ethyl)-1H-imidazole |...)
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM21392(3-(2-aminoethyl)-1H-indole-5-carboxamide | 5-CT | ...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM22904((2R)-1-(1H-imidazol-5-yl)propan-2-amine | (R)-alph...)
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM22911(2-(3H-imidazol-4-yl)ethylsulfanylmethanimidamide |...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Homo sapiens (Human))
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.590nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.780nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317868(4-(2-(4-tert-Butylphenylamino)ethyl)-1H-imidazole ...)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.950nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317864(4-(2-(4-Trifluoromethylphenylamino)ethyl)-1H-imida...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317865(2-(2-(4-tert-Butylphenylthio)ethyl)-1H-imidazole |...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of human recombinant histamine H4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataKi:  1.33nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1a receptor(RAT)
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  1.45nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403759(CHEMBL428494)
Affinity DataKi:  1.90nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403759(CHEMBL428494)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220557(CHEMBL422869)
Affinity DataKi:  2nMAssay Description:Ability to displace the radioligand [3H]5-carboximidotryptamine ([3H]-5-CT) from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-(4-(4-phenyl-5,6-dihydropyridin-1(2H)-yl)butyl)...)
Affinity DataKi:  2.10nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-(4-(4-phenyl-5,6-dihydropyridin-1(2H)-yl)butyl)...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50116963(2a-(4-(4-phenyl-5,6-dihydropyridin-1(2H)-yl)butyl)...)
Affinity DataKi:  2.10nMAssay Description:Ability to displace the radioligand [3H]5-carboximidotryptamine ([3H]-5-CT) from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM86039(DR4004)
Affinity DataKi:  2.14nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317867(4-(2-(3-tert-Butylphenylamino)ethyl)-1H-imidazole ...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50473640(CHEMBL71847)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403770(CHEMBL12427)
Affinity DataKi:  3.30nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403770(CHEMBL12427)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220558(CHEMBL418888)
Affinity DataKi:  3.5nMAssay Description:Ability to displace the radioligand [3H]5-carboximidotryptamine ([3H]-5-CT) from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220558(CHEMBL418888)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403768(CHEMBL273246)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403768(CHEMBL273246)
Affinity DataKi:  3.80nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403780(CHEMBL12846)
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317866(4-(2-(4-Cyclohexylphenylamino)ethyl)-1H-imidazole ...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50473633(CHEMBL304731)
Affinity DataKi:  4.80nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220504(CHEMBL348410)
Affinity DataKi:  5nMAssay Description:Ability to displace the radioligand [3H]5-carboximidotryptamine ([3H]-5-CT) from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403777(CHEMBL12702)
Affinity DataKi:  5.10nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403777(CHEMBL12702)
Affinity DataKi:  5.10nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50130272(2a-[3-(4-Phenyl-piperazin-1-yl)-propyl]-2a,3,4,5-t...)
Affinity DataKi:  5.20nMAssay Description:Compound was evaluated for its ability to displace [3H]5-CT binding from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSerotonin 2 (5-HT2) receptor(RAT)
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50403772(CHEMBL268921)
Affinity DataKi:  5.40nMAssay Description:Compound was evaluated for its ability to displace [3H]ketanserin binding from cloned rat cerebral cortex membranes 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50473658(CHEMBL71383)
Affinity DataKi:  5.80nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50473644(CHEMBL302766)
Affinity DataKi:  6nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  6.36nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50473648(CHEMBL71225)
Affinity DataKi:  6.5nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50473651(CHEMBL71959)
Affinity DataKi:  7.10nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi:  7.20nMAssay Description:Ability to displace the radioligand [3H]5-carboximidotryptamine ([3H]-5-CT) from cloned human 5-hydroxytryptamine 7 receptor expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50220503(CHEMBL348890)
Affinity DataKi:  7.20nMAssay Description:Binding affinity towards 5-HT7 receptor by the displacement of [3H]-5-CT] in human recombinant receptors in mammalian cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50473639(CHEMBL303166)
Affinity DataKi:  7.90nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50473652(CHEMBL422587)
Affinity DataKi:  8.10nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50473657(CHEMBL70889)
Affinity DataKi:  8.70nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute of New Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  9.42nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Meiji Seika Kaisha

Curated by ChEMBL
LigandPNGBDBM50317869(4-(2-(3,4-Dimethylphenylamino)ethyl)-1H-imidazole ...)
Affinity DataKi:  9.90nMAssay Description:Displacement of [3H[N-alpha-methylhistamine form human recombinant histamine H3 receptor expressed in CHO cells after 1 hr by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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